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5-(2,5-difluorobenzoyl)-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(3-methylpyridin-2-yl)-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
3-chloro-N-(2-hydroxypropyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-(6-methoxynaphthalene-2-carbonyl)-1-(1-propylpiperidin-4-yl)piperidine
2-fluoro-4-({[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}methyl)-6-methoxyphenol
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
(2S,4R)-4-(cycloheptylamino)-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3aS,6aR)-3-cyclopentyl-5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-methoxy-9-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
1-(1-{[4-(phenylamino)quinazolin-2-yl]methyl}piperidin-4-yl)propan-1-ol
2-[4-(4-{[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]amino}piperidin-1-yl)phenyl]-N-[2-(3-fluorophenyl)ethyl]acetamide
1-cyclopropyl-4-({[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)pyrrolidin-2-one
3-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-5-(propan-2-yl)-1,2-oxazole
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
3-(1H-indazol-5-yl)-1-{[1-(2-phenylethyl)piperidin-4-yl]methyl}urea
4-[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-sulfonamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-{[3-(1-methyl-1H-pyrazol-4-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(1-ethylpiperidin-4-yl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(2-methylpyridin-4-yl)methyl]quinoline-4-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
1-[1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
1-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azetidin-3-yl)-2-methylpiperidine
(2E)-3-(2-chlorophenyl)-N-cyclopropyl-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)prop-2-enamide
N-cyclopropyl-3-(3-fluorophenyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
5-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2,6-dimethylpyrimidine
2-phenyl-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
N-[(3R,4S)-1-(1-cyclopropanecarbonylpiperidin-4-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-methylpropyl)acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
N-(3,3-dimethylcyclohexyl)-1-methanesulfonylpiperidin-4-amine
N-(1H-imidazol-2-ylmethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
3-(2-{[6-(methoxymethyl)pyrimidin-4-yl]amino}ethyl)-1,3-oxazolidin-2-one
(2R,3S,6R)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-5-(methoxymethyl)-1,3,4-oxadiazole
2-{[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]methyl}-3-methylquinoxaline
5-ethyl-6-methyl-N4-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}pyrimidine-2,4-diamine
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(2,2-dimethyloxan-4-yl)pyridin-2-amine
2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-N,N-dimethylethane-1-sulfonamide
3-{5-[1-(4-methoxyphenyl)cyclopropyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
1-[(6-methylpyridin-2-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]benzonitrile