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(3S)-1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-ol
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-propoxypiperidine
N-cyclopentyl-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
8-[(6-methylpyridin-2-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(3-{[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-4-methoxyphenyl)acetic acid
4-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}pyridine
(3S,4S)-1-(azetidine-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
methyl (2S,4R)-4-[3-(3-fluorophenyl)benzamido]-1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidine-2-carboxylate
(4aS,8aR)-6-(5-methyl-1,2-oxazole-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-1,2-oxazole
2-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)-6-methylphenol
7-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(5-chloro-2-methoxyphenyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[4-({[(3S)-1-benzylpyrrolidin-3-yl]carbamoyl}methoxy)phenyl]propanamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
4-[1-(2-fluoro-5-sulfamoylphenyl)-5-methyl-1H-1,2,4-triazol-3-yl]benzamide
N-[4-(3-methylphenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N'-cycloheptyl-N-(2-hydroxy-3-phenylpropyl)butanediamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-{1-[(3,4,5-trimethoxyphenyl)methyl]-1H-imidazol-2-yl}benzonitrile
N-(3,3-diphenylpropyl)-6-(furan-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(3,5-dimethylfuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-methoxypropanamide
2-(2,6-difluorophenyl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
3-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[(3R,4S)-4-cyclopropyl-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]-3,3,3-trifluoropropanamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
7-(cyclopropylmethyl)-2-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-(3-fluorophenoxy)-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine-4-carboxylic acid
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)(oxolan-2-ylmethyl)amine
N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)cyclopentanecarboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
5-[(2-fluorophenyl)methyl]-3-(oxan-4-ylmethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-(4-methoxyphenoxy)-1-(thiophene-3-carbonyl)piperidine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(2H-1,2,3-benzotriazol-2-yl)acetamide
[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
N,N-diethyl-2-{4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1H-1,2,3-triazol-1-yl}acetamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[3-(methylsulfanyl)propyl]-1,3-benzoxazole-6-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
methyl 2-(4-hydroxyphenyl)-1H-1,3-benzodiazole-6-carboxylate
4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-5-one
3-(1H-imidazol-2-yl)-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]benzamide
N-(pyridin-2-ylmethyl)-4-{thieno[3,2-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
4-fluoro-N-(3-{4-[methyl(oxolan-3-yl)amino]piperidin-1-yl}phenyl)benzene-1-sulfonamide
2-cyclopropyl-1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
N-ethyl-4-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
methyl 6-[(2-hydroxyphenyl)methyl]-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide