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4-{[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl}){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-{1-[1-(1-carbamoylethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
cyclopentyl 4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}amino)benzoate
ethyl 4-({1-[4-(2-fluorobenzamido)phenyl]piperidin-4-yl}amino)piperidine-1-carboxylate
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(3-methoxybenzoyl)piperazine
1-(cyclopropylmethyl)-5-[3-(dimethylamino)benzoyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
propan-2-yl 4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxylate
4-{1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl}benzoic acid
1-[2-(3-fluorophenyl)ethyl]-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-6-oxopiperidine-3-carboxamide
1,7-dimethyl-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
(4-{[3-(4-methylpiperazin-1-yl)propyl]amino}quinazolin-2-yl)methanol
N-cyclopentyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N,N-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
4-({1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2,5-dimethylpyrazine
(1R,7S)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-phenyl-4-(3-phenylbutanoyl)piperazin-2-one
2-(2-aminoethyl)-N-[1-(3,4,5-trimethoxyphenyl)ethyl]quinazolin-4-amine
1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]sulfamoyl}dimethylamine
1-(cyclohexylmethyl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-methylpropyl)-2-(pyridin-2-yl)-N-(pyridin-2-ylmethyl)acetamide
(5-{[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
N-[1-(1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)ethyl]-N-methylacetamide
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]acetamide
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(thian-4-yl)piperazine
(4aS,7aR)-1-[(2-methylpyrimidin-5-yl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,5R,6S,7aS)-2-[(1-benzyl-1H-imidazol-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
3-[(3R,4S)-1-(2-methyl-1,3-benzothiazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(2-propylpyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
methyl 4-[5-({4-[(4-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
1-{2-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
(2S,4S)-4-amino-N-[(5-chloro-2-methoxyphenyl)methyl]-N,1-dimethylpyrrolidine-2-carboxamide
3-chloro-2-(4-methanesulfonylphenyl)-5-methylpyridine
4-chloro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
methyl 2-(3-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}-1H-indol-1-yl)acetate
(2R,3S,6R)-5-cyclobutanecarbonyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,7S)-3-[2-(4-methylphenyl)ethyl]-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-[(4-chlorophenyl)methyl]-6-oxo-N-[3-(pyridin-3-yloxy)propyl]piperidine-3-carboxamide
(2S,4R)-1-[(3-methoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(piperidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,6R)-9-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one