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N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
2-(cyclohex-1-en-1-yl)-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)acetamide
2-[(3,4-dimethoxypyridin-2-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N,N-dimethyl-5-[3-(1H-pyrazol-1-yl)phenyl]pyridin-2-amine
3,5-dichloro-4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}pyridine
3-[4-(quinolin-6-yl)-1H-pyrazol-1-yl]propanamide
2-{5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
(2-{2-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
methyl 4-{2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetamido}butanoate
N-(1-cycloheptylpiperidin-3-yl)-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
2-{2-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
ethyl 3-{[5-(tert-butylcarbamoyl)-1-cyclohexyl-4-oxo-1,4-dihydropyridin-3-yl]formamido}propanoate
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2-(1H-pyrazol-1-yl)butanamide
1-[3-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-1-yl]propan-1-one
3-(2-methyl-1H-imidazol-1-yl)-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazine
(1R,5S,8S)-N-(3,5-dichlorophenyl)-8-hydroxy-3-azabicyclo[3.2.1]octane-3-carboxamide
[3-(3-methylbut-2-en-1-yl)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]methanol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]propan-1-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethan-1-one
4-[3-(azepane-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazine-1-carbaldehyde
4-(3-chloropyridin-4-yl)-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
(2R,3R)-3-amino-1'-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-cyclopropyl-1-ethyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazole
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazine
2-{[(4-acetylphenyl)carbamoyl]amino}-N,N,3-trimethylbutanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]butan-1-one
2-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}pyridine-4-carbonitrile
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(1,3-thiazol-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(3-cyanophenyl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
2-methyl-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-octahydro-1H-pyrazino[1,2-a]piperazine
ethyl 4-[6-(2,1,3-benzothiadiazol-5-ylmethyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
3-fluoro-N-[(3-methoxyphenyl)methyl]-5-methyl-N-(prop-2-en-1-yl)imidazo[1,2-a]pyridine-2-carboxamide
4-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-N-[2-(methylsulfanyl)phenyl]-4-oxobutanamide
(1H-imidazol-2-ylmethyl)(methyl){[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}amine
(2S)-2-acetamido-N,4-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pentanamide
2-(2-methoxy-4-methylphenoxymethyl)-4-(pyrrolidine-1-carbonyl)-1,3-oxazole
5-[1-(2-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]pyridin-2-amine
1-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
(2E)-N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2-methoxy-2-methylpropyl)piperidine-3-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
(5S,9aS,9bS)-5-(3,5-dimethyl-1H-indol-2-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2-{1-[(6-chloropyridin-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one
2-{[3-(methylsulfanyl)phenyl]methyl}-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine