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3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-[(1S)-2-hydroxy-1-phenylethyl]urea
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
5-(4-acetylphenoxymethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
3-[2-(dimethylsulfamoyl)ethyl]-1-(1-ethyl-1H-1,2,3-triazol-4-yl)urea
(4aS,8aR)-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-(3-methylthiophen-2-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
2-(2-methoxyethyl)-6-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,3-benzoxazole
N-{1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-4-yl}acetamide
3-({1-[2-(dimethylamino)acetyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carboxamide
N-(1H-indol-2-ylmethyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
(2S)-2-amino-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pentan-1-one
9-[3-(3-fluorophenyl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-N-[4-(oxolan-2-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
2-(4-methoxy-3-methylphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
8-methoxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-amino-1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
1-{4-[3-(morpholin-4-ylmethyl)phenyl]phenyl}ethan-1-ol
N-(4-{4-[(1-benzylpiperidin-3-yl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
ethyl 2-(1-{3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxyphenyl}-N-methylformamido)acetate
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,4-diazepane
(3R,4R)-3-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(oxan-4-yl)piperidin-4-ol
3-(3,6-dimethylpyrazin-2-yl)-5-methyl-1H-indole
N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
6-methyl-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]quinoline
1-[3-(3-methoxyphenyl)phenyl]-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-6-(2,4,6-trimethylphenyl)pyrimidin-4-amine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
(3aR,6aS)-5-[3-(dimethylamino)-2,2-dimethylpropyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-amino-6-(4-ethylphenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-(dimethylamino)propan-2-ol
(2S)-1-acetyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N,1-dimethyl-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(pent-4-enoyl)pyrrolidine-2-carboxamide
8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methylthiophen-2-yl)methyl]piperidine
4-fluoro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
(3R,5S)-5-(3-fluorophenoxymethyl)-1-[(4-hydroxyphenyl)methyl]-N-[2-(morpholin-4-yl)ethyl]piperidine-3-carboxamide
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-(5-methylfuran-2-yl)-1H-pyrazole
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
N-(4-methoxy-3,5-dimethylphenyl)thiomorpholine-4-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
5-ethyl-4-({3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}methyl)furan-2-carboxamide
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
1-{3,5-dimethyl-4-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one