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1-(3-methoxyphenyl)-4-{3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanoyl}piperazin-2-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}acetic acid
(1R,5S,8S)-8-methoxy-N-[4-(propylsulfamoyl)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
N-(2-fluoroethyl)-3-{[1-(pyridin-4-yl)propan-2-yl]sulfamoyl}benzamide
N-cyclopentyl-5-[2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
5-cyclopropanecarbonyl-1'-(2-phenylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[2-(pyridin-4-ylsulfanyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
1-methyl-1'-(morpholine-2-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-cyclobutyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-phenyl-1-[1-(quinoxaline-5-carbonyl)piperidin-4-yl]ethan-1-ol
6-[6-hydroxy-4-(1H-imidazol-4-ylmethyl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
2-{1-[(2-ethoxyphenyl)methyl]-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl}ethan-1-ol
4-(2-{4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-1-yl}ethyl)morpholine
2-{2-[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]ethoxy}ethan-1-ol
4-(1H-pyrazol-4-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
(3S,4R)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-3-methylthiophene-2-carboxamide
1-[2-(diethylamino)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-{2-[4-(diphenylmethyl)piperazin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}phenol
(1R,9aR)-1-{1H-pyrrolo[2,3-b]pyridin-1-ylmethyl}-octahydro-1H-quinolizin-1-ol
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]acetamide
2-[4-(cyclopropanesulfonyl)morpholin-3-yl]-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]acetamide
3-[5-(3-methoxypropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
1-{1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
7-[(3-methoxyphenyl)methyl]-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decane
4-hydroxy-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methylpyrimidine-5-carboxamide
N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]oxolane-3-carboxamide
3-(isoquinolin-5-yl)-5-(morpholine-4-sulfonyl)benzoic acid
2-{[2-(ethoxymethyl)-7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
N-(1-benzothiophen-2-ylmethyl)-2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
2-(3-fluorophenyl)-5-[2-(methylsulfanyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
8-[(2E)-3-phenylprop-2-en-1-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(4aS,7aR)-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}pyridine
1-(3-methoxypropyl)-3-(2-oxo-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethyl)-3-phenylpyrrolidine-2,5-dione
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
3-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridazine
5-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
1-(pyrrolidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}cyclopentane-1-carboxamide
(4aS,8aR)-6-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(cyclohex-1-ene-1-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
5-[3-(4-methylphenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-(4-acetylphenyl)-1-benzyl-1-(4-hydroxybutyl)urea
2-(2-ethyl-1H-imidazol-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide