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2-[(3-fluorophenyl)methyl]-N-(2-methoxyethyl)-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
2-{1-[3-(2-methylphenyl)propyl]pyrrolidin-2-yl}pyridine
1-{[4-({3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenyl]methyl}-1H-pyrazole
N-(1-hydroxypropan-2-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-(4-methoxyphenoxymethyl)-4-(3-propylpyrrolidine-1-carbonyl)-1,3-oxazole
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(methylsulfanyl)ethyl]propanamide
7-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
1'-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2,4-dimethoxyphenyl)methyl]methylamine
2-chloro-4-{2-[2-(dimethylamino)ethoxy]phenyl}benzamide
4-(1-phenylmethanesulfonylpiperidin-3-yl)morpholine
7-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-1-oxa-7-azaspiro[3.5]nonane
4-cyclobutyl-6-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]pyrimidin-2-amine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-fluorobenzamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
methyl 3-benzamido-5-{[(3-fluorophenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-benzyl-1-({4-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)piperidine
2-{1-[(2-fluorophenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-{4-[4-(dimethylamino)phenyl]-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl}methanesulfonamide
2-[ethyl(methyl)amino]-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
1-(4-methylphenyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazin-2-one
N,N-dimethyl-2-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-amine
(4aR,8aR)-4-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-octahydro-2H-1,4-benzoxazine
1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}urea
4-[3-(1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyridine
2-[4-(1-benzofuran-2-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[3-(dimethylamino)propyl]-9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]-1-(pyrrolidin-1-yl)ethan-1-one
N-[(3S,4R)-1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
6-(1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)-2-methyl-3,4-dihydropyrimidin-4-one
N-benzyl-5-{[(5-chlorothiophen-2-yl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
2-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
5-chloro-6-[3-(hydroxymethyl)phenyl]-2-methylpyrimidin-4-ol
1-[(1-{6-[(2-hydroxybutyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3,4,5-trimethoxyphenyl)urea
N,N-diethyl-1-(3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanoyl)piperidine-3-carboxamide
N-[2-(2-ethoxyethoxy)phenyl]-2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
4-(2-phenylethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
methyl 8-[3-(furan-2-yl)benzoyl]-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(1,2,3,4-tetrahydronaphthalen-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3-(propoxymethyl)pyrrolidine
1-(3-ethoxybenzoyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine