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N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
5-(1H-indazol-1-yl)pyridin-2-amine
4-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-2-ethylpyrimidine
N-methyl-N-({5-[(3-phenylpiperidin-1-yl)methyl]furan-2-yl}methyl)methanesulfonamide
2-butyl-8-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-fluoro-2-methylphenyl)methyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-(1H-imidazol-2-ylmethyl)-3-methylurea
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-1'-[4-(1H-pyrazol-3-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,3S)-7-[3-(dimethylamino)benzoyl]-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
1-{3-[2-(azetidin-1-ylmethyl)phenoxy]propyl}piperidine
1-{2-[3-(4-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methoxy-4-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]phenol
{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1-methylpiperazin-2-yl}methanol
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-pyrazole-3-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(4-methoxyphenyl)methyl]piperidine
{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-4-ylmethyl)amine
ethyl 3-{[(1-cycloheptylpiperidin-3-yl)carbamoyl]amino}propanoate
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-7-[(2-methyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,N-dimethyl-2-[(1S,5R)-6-(4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-ethyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-cyclopropyl-1-[1-(quinoxalin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-N-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}propanamide
(1R,5R)-N,N-dimethyl-6-[2-(pyridin-2-ylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-ethyl-N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2R,3S,6R)-5-[(5-ethylfuran-2-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
{[4-(methylsulfanyl)phenyl]methyl}({[2-(propan-2-yl)pyrimidin-4-yl]methyl})propylamine
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3-propylpiperidine-3-carboxylic acid
8-{5-[(methylsulfanyl)methyl]pyridin-2-yl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-methyl-N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}benzamide
2-(2-fluorophenyl)-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-4-(pyridin-3-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrimidin-2-amine
(4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}morpholin-2-yl)methanamine
2-(3,4-dimethoxyphenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
ethyl 1-(1-benzofuran-2-carbonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
1-{3-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]propyl}-6-methyl-1,2-dihydropyridin-2-one
5-(naphthalen-2-yl)-3-[2-(pyridin-2-yl)pyrrolidin-1-yl]-1,2,4-triazine
1-[2-(dimethylamino)-6-[3-(methylsulfanyl)propyl]-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
4-{[3-(3-methoxyphenoxymethyl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-{1-[2-(dimethylamino)benzoyl]piperidin-4-yl}piperidin-3-ol
6-cyano-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
2-amino-4-(2,5-difluorophenyl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-ethyl-5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1H-indole
4-[4-(methylsulfanyl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine