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7-(cyclohexylmethyl)-2-[(2-ethylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-{3-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidin-1-yl}pyridine
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
5-(1H-1,3-benzodiazol-2-ylmethyl)-N-benzyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-methoxypropan-2-yl)-7-(thiophene-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 2-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxylate
1-[(5-methylthiophen-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-[3-(3-methylphenyl)propyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-benzyl-N-ethyl-1,3-oxazole-4-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
8-(quinoline-6-carbonyl)-1-oxa-8-azaspiro[4.5]decane
3-(2-chlorophenyl)-N-[(methylcarbamoyl)methyl]-3-phenylpropanamide
2-(3,4-dichlorophenyl)-4-{furo[3,2-c]pyridin-4-yl}morpholine
N-{3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]phenyl}propanamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-methoxyacetamide
2-{5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}-6-methylpyridine
5-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-4-(pyrimidin-2-ylsulfanyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-chloro-2-methyl-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzene-1-sulfonamide
2-methyl-4-{3-[1-(pyrrolidin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
dimethyl[(4-{[3-(2-methylphenyl)phenyl]methyl}-1,4-oxazepan-6-yl)methyl]amine
1-({5-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)azepane
2-[3-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-4-(propan-2-yl)-1,3-thiazole
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-4-methoxy-N-[(4-methoxyphenyl)methyl]benzamide
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]oxane-2-carboxamide
N-ethyl-N-[2-(3-ethylphenoxy)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
1,6-dimethyl-3-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
methyl N-{[(2S,4S)-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-4-fluoropyrrolidin-2-yl]methyl}carbamate
3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]-1-(thiomorpholin-4-yl)propan-1-one
(butan-2-yl)({imidazo[1,2-a]pyrimidin-6-ylmethyl})(3-phenylprop-2-yn-1-yl)amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[1-(2-phenylethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
3-methyl-4-{1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-1,2,5-oxadiazole
2-{4-[(3-chloro-4-methoxyphenyl)methyl]morpholin-2-yl}ethan-1-ol
N-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
1-{2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
8-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2,4-dimethyl-N-[2-(3-methylphenyl)-1,3-benzoxazol-6-yl]-1,4-diazepane-1-carboxamide
1-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-methylpropan-1-one
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]propanamide
2-(pyridin-4-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-methyl-7-[2-(morpholin-4-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-amino-5-ethyl-4-(4-hydroxy-3-methoxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
[(3R,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(5-ethylpyridin-2-yl)methyl]-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide