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N-[(3S,4R)-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
{1-[(2-aminopyrimidin-5-yl)methyl]-3-propylpiperidin-3-yl}methanol
5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-benzyl-4-methylpiperidin-4-ol
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(1-phenylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-(pyridin-4-ylmethyl)acetamide
2-[(3-fluorophenyl)methyl]-4-[2-(methylsulfanyl)benzoyl]morpholine
3-{[2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)acetamido]methyl}-4-methylbenzoic acid
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
4-ethenyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}benzamide
N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinoline-6-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
2-methyl-4-(4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}phenyl)butan-2-ol
2,5-dimethyl-3-(4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)pyrazine
4-cyclopentyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
1-(6-aminopyridine-3-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
{3-[(3-methoxyphenyl)methyl]-1-[(4-methoxyphenyl)methyl]piperidin-3-yl}methanol
N-[2-(2-chlorophenyl)-1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)ethyl]-N-methylfuran-2-carboxamide
9-(5-chloro-2-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-yl)pyridine
3-methyl-4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazin-2-one
2-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(2-fluorophenyl)methyl]-N-propylacetamide
N-(cyclopropylmethyl)-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[(3-{2-[1-(3-fluorobenzoyl)piperidin-2-yl]ethoxy}-4-methoxyphenyl)methyl]morpholine
N-(oxan-4-yl)-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
1-(1,3-benzothiazol-5-yl)-3-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}urea
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylthiophene-2-carboxamide
2-{[3-(4-fluorophenoxy)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
4-(2,2-diethylmorpholine-4-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
2-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-1,2,3,4-tetrahydroisoquinoline
4-(2-methyl-1-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}propan-2-yl)morpholine
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-methanesulfonylpiperidin-3-yl)propanamide
ethyl 4-[6-amino-2-(diethylamino)pyrimidin-4-yl]piperazine-1-carboxylate
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-{7-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3-methoxypropanamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-phenoxypropan-1-one
ethyl 2-(4-methanesulfonylphenyl)pyridine-3-carboxylate
8-(furan-3-ylmethyl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-ethoxy-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
N,N-dimethyl-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]azepan-4-amine
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[(5-ethylpyridin-2-yl)methyl]-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
(2S,3R)-2-({[(3,5-dimethoxyphenyl)carbamoyl]methyl}amino)-3-hydroxybutanamide
2-[4-(2,2-dimethylpropyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol