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3-{[(2,1,3-benzothiadiazol-5-ylmethyl)amino]methyl}-5-acetamido-N-(2-methoxyphenyl)benzamide
4-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
(2E)-4-methyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-2-enamide
4-[2-(3-fluorophenyl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
3-[(methylsulfanyl)methyl]-N-{4-[(trifluoromethyl)sulfanyl]phenyl}piperidine-1-carboxamide
6-(methoxymethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}pyridine-2-carboxamide
3-(but-3-en-1-yl)-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-{3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(6-methoxy-1H-indazol-3-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-methyl-6-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
(3R,4S)-4-cyclopropyl-1-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}pyrrolidin-3-amine
2-butyl-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}-2,5-dihydro-1H-pyrrole
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(4-benzylpiperazin-1-yl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
1-[4-({[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-{1-[2-(tert-butylcarbamoyl)ethyl]piperidin-3-yl}benzoic acid
N-(adamantan-1-ylmethyl)-1-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-(benzylamino)-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(dimethylamino)-N-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(2-methylphenyl)acetamide
1-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-4-yl}piperidin-4-ol
4-(1H-indol-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]butanamide
2-{[6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}acetamide
N-[(1-methylpiperidin-4-yl)methyl]-3-(methylsulfanyl)propanamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepane
2-[3-(methoxymethyl)phenyl]-2-[methyl(pyridin-3-ylmethyl)amino]acetic acid
3-(3-fluoro-4-methoxyphenyl)-4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(2-methylphenyl)-1H-pyrazole
1-[5-(3-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)thiophen-2-yl]ethan-1-one
1-methyl-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
6-({[(4-phenylphenyl)methyl]amino}methyl)-1,4-oxazepan-6-ol
3-(propan-2-yl)-5-[4-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazole
N-ethyl-1-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
5-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-3-(4-methoxyphenyl)-1H-pyrazole
3-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanoic acid
4-(2-hydroxypropan-2-yl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
7-(2-methylphenyl)-4-(6-methylpyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
1-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)methyl]-4-(3-methylpyridin-4-yl)piperazine
6-methyl-N4-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidine-2,4-diamine
5-{[4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazol-2-yl]methoxy}isoquinoline
3-[(3R,4S)-1-(5-cyano-4,6-dimethylpyridin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-{3-[(3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-pyrazol-5-yl)methoxy]phenyl}ethan-1-one
1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine
2-(4-methyl-1,4-diazepan-1-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-(4-chlorophenyl)-N-({1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide