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[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-methylbenzamide
1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}azocane
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(3-methoxypropyl)piperidine
5-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1,3-oxazole
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[(4-phenyloxan-4-yl)methyl]propanamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-(4H-1,2,4-triazol-3-ylmethyl)piperazine
2-(4-acetylphenoxy)-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
7-fluoro-2-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}quinoline-4-carboxamide
8-chloro-2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}quinolin-4-ol
N-benzyl-N-methyl-3-({[3-(morpholin-4-yl)propyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
4-[2-(2-chlorophenyl)ethyl]-11-[(prop-2-en-1-yl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-(4-methylpiperazin-1-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
methyl (2S,4R)-4-(dimethylamino)-1-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxylate
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N3-butyl-N5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-butyl-3-(furan-2-yl)-5-(oxan-4-yl)-1H-1,2,4-triazole
2-(methoxymethyl)-5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrimidine
1-benzyl-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(3-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
2-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)furan-3-carboxamide
methyl 4-{4-[2-(ethylamino)pyrimidine-5-carbonyl]piperazin-1-yl}benzoate
5-(2,6-dimethylphenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-{1-[(3-chlorophenyl)methyl]-5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl}pyridine
N-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}-2-(pyrrolidin-3-yl)benzamide
1-(1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
3-(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-1-benzyl-N-methyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-methyl-4-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-cyclopentyl-N-(3-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[2-(ethanesulfonyl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[(3S,4R)-1-[1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]-4-propylpyrrolidin-3-yl]acetamide
1-(2-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-4-(piperidin-1-ylmethyl)benzamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
2-{4-chloro-2-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]phenoxy}acetamide
N-[2-(pyridin-4-yl)ethyl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
(2R)-2-amino-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-(2-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)carbamoyl]amino}phenyl)-N-methylpropanamide
3-cyclopropyl-5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-fluoro-3,5-dimethylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-(3-fluorophenyl)-1H-pyrazole
(3R,4R)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol