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N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
(1S,5R)-3-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
1-(2-methylphenyl)-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
methyl 3-({imidazo[2,1-b][1,3]thiazol-6-ylformamido}methyl)-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate
1-[4-({[(3-chlorophenyl)methyl](methyl)amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[2-(1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
2-(4-fluoro-2-methylphenyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
5-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-butyl-4-[2-(4-ethyl-1,4-diazepan-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
2-(dimethylamino)-N-(3-hydroxy-3-methylbutyl)-N-methyl-2-(3-methylphenyl)acetamide
N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-[2-methyl-3-(pyrrolidin-1-yl)propyl]propanamide
(2S)-2-(methoxymethyl)-1-[2-(4-methoxyphenoxy)ethyl]pyrrolidine
1-cyclopentanecarbonyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
8-[(2-fluoro-5-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
3-(2-propoxybenzoyl)-3,9-diazaspiro[5.6]dodecan-10-one
4-(2-fluorobenzenesulfonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
N,N-dimethyl-3-{4-[({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}carbamoyl)amino]phenyl}propanamide
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
N-[(3S,4R)-1-[(3-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-(4-{4-azaspiro[2.5]octan-4-ylmethyl}-2-methoxyphenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]acetamide
3-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-dihydrophthalazin-1-one
4-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-3-yl}morpholine
8-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}quinoline
N-[(2S)-2-aminopropyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-(3-hydroxypropyl)-1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidine-3-carboxamide
3-[ethyl({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
1,3-dimethyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-N-(2,5-dimethoxyphenyl)-3-oxopropanamide
3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-methylpropanamide
3-benzyl-4-(2-methylquinoline-4-carbonyl)piperazin-2-one
(5-{2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-1H-1,3-benzodiazol-2-yl)methanol
{4-[(4-methoxyphenyl)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}methanol
1-ethyl-5-{4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazol-5-yl}-1H-1,2,4-triazole
3-{5-[2-(trifluoromethyl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-[3-(1H-imidazol-1-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-benzyl-3-[3-(pyridin-3-yl)propyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-[1'-(2-cyclopentylacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(3S,4R)-4-(4-methylphenyl)-1-(2,4,5-trimethylbenzoyl)pyrrolidin-3-yl]acetamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-(2-chloropyridine-4-carbonyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine