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(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-methyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-(thiophene-2-sulfonyl)piperidine
1-(2,4-dimethoxybenzenesulfonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
3-benzyl-4-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]piperazin-2-one
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
4-({[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-methoxyphenol
5-[(2-ethyl-4-methyl-1H-imidazol-1-yl)methyl]-3-(thiophen-2-yl)-1,2,4-oxadiazole
2-(4-fluorophenyl)-2-hydroxy-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{4-[(2,4-difluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2,2-diethyl-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)cyclopropane-1-carboxamide
3-{[1-(2,2-difluorocyclopropanecarbonyl)piperidin-4-yl]methyl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N1-(prop-2-en-1-yl)-N2-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1,2-dicarboxamide
1-(2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanamine
2-[3-(2,5-dimethylfuran-3-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-fluoro-N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}benzamide
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-4-propylpyrimidine
8-chloro-2-(furan-2-yl)-N-(oxan-4-yl)quinoline-4-carboxamide
methyl 4-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butanoate
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(quinolin-4-ylmethyl)amine
2-[3-(2-methoxyethyl)-5-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-[2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(pyridin-3-yloxy)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-benzothiazole
6-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-N-methylpyridin-2-amine
N-cyclopropyl-6-ethyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(thiophene-2-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
5-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
4-hydroxy-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[(4-methoxyphenyl)methyl]-4-(4-methyl-1,3-oxazole-5-carbonyl)morpholine
3-({1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](isoquinolin-5-ylmethyl)methylamine
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[1-(pyridin-4-yl)propyl]benzamide
1-methyl-8-{2-[4-(methylsulfanyl)phenyl]acetyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-N-(3-phenylprop-2-yn-1-yl)cyclopropanamine
N-[(2R,3R)-1'-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
ethyl 1-cyclopentanecarbonyl-4-(3-phenylpropyl)piperidine-4-carboxylate
(4S,4aS,8aS)-1-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]-4-phenyl-decahydroquinolin-4-ol
methyl 6-[(4-ethylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aS,7aR)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
8-(isoquinolin-5-ylmethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-methyl-1-[3-(1,3-oxazol-5-yl)phenyl]-3-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one