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N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-4-methyl-1,3-thiazole-5-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
1-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2,4,6-trifluorophenyl)ethan-1-one
3-(4-chloro-2-methylbenzoyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3-(1H-pyrazol-5-yl)piperidine
5-cyclobutanecarbonyl-1'-(1-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3,5-dimethylphenyl)-N-[(3,4,5-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-phenyl-N-[1-(pyridin-3-ylmethyl)azepan-4-yl]-1,2-oxazole-4-carboxamide
4-(1H-imidazol-2-ylmethyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-(2-chlorophenyl)-3-{1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
5-(4-chlorobenzoyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(3-chloro-4-fluorophenyl)-4-{1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}pyridine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-(2-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
N-[1-({[(3S)-2-oxoazepan-3-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
3-(ethylamino)-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
4-[2-(benzenesulfonyl)ethyl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
ethyl 4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
(1R,5R)-6-(cyclobutylmethyl)-3-{imidazo[1,2-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
2-(ethylsulfanyl)-5-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
3-(3-methoxyphenyl)-5-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-(2-{[methyl(propyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)propanoic acid
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
4-[(2,4-dichlorophenyl)methyl]-3-(dimethyl-1,3-oxazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
(2R,4R)-N-[(2,3-dimethoxyphenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
4-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-[2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]-6-phenyl-2,3-dihydropyridazin-3-one
(3aS,6aR)-5-[(3-fluoro-4-methoxyphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-cyclopropyl-6-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
(4aS,8aR)-6-(1,3-oxazole-4-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[6-hydroxy-4-(2-phenylquinolin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(pyrrolidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(benzyloxy)azetidine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
2-chloro-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]pyridine-4-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
ethyl 1-(3,3-dimethylcyclohexyl)-4-(2-methoxyethyl)piperidine-4-carboxylate
5-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-N,N-dimethylpyridin-2-amine
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
N-(2,4-dimethylphenyl)-2-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}acetamide
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-ethyl-1H-pyrazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-ethyl-5-({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-(3,3-diphenylpiperidine-1-carbonyl)-1-(propan-2-yl)pyrrolidin-2-one
(1s,4s)-4-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]cyclohexan-1-ol
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
3-{3-[cyclohexyl(methyl)amino]propyl}-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(3-propyl-1,2,4-oxadiazol-5-yl)phenyl]imidazolidin-2-one