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1-(dimethyl-1,3-oxazole-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-butoxy-1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}ethan-1-one
N-[(3R,4S)-1-(4,6-dimethylpyrimidin-2-yl)-4-propylpyrrolidin-3-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
3-[(methylsulfanyl)methyl]-5-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
N-benzyl-5-{[(4-methoxyphenyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{5-[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
3-{2-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
7-(propan-2-yl)-2-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(1H-pyrazol-4-yl)-5-(trifluoromethyl)pyridine
N-methyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]ethyl}thiophene-3-carboxamide
3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(methoxymethyl)-1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidine
5-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-cyclopropyl-3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(2-methoxyphenyl)methyl]propanamide
1-(2-chlorophenyl)-3-(1-{1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
1-[(4-methanesulfonylphenyl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
2-{6-chloro-3-[(3,4-dimethylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-[4-(4-chlorophenoxy)piperidine-1-carbonyl]benzonitrile
{[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl}(propan-2-yl)amine
1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-{[4-(5-chlorothiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(prop-2-en-1-yl)-1H-pyrazole
propyl 4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-(2-methylphenoxy)azetidine
(2R,3R)-3-[methyl(propyl)amino]-1'-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(1S,5R)-6-benzyl-3-[2-(3-oxopiperazin-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(3,4-difluorobenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
6-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-butyl-2-cyclobutaneamido-N-methyl-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2,7-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-(3-methylphenoxy)piperidine
2-(cyclopropylmethyl)-7-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}oxy)pyridine
2-(dimethylamino)-N-[3-(dimethylamino)propyl]-2-(3-fluorophenyl)acetamide
(1S,5R)-6-[(5-methylthiophen-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-hydroxy-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(4aR,7aS)-1-methyl-4-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)pentanoate
N-(3,4-dimethyl-1H-pyrazol-5-yl)-2-[4-(methylsulfanyl)phenyl]acetamide
8-[4-(piperidin-1-ylmethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,7aR)-4-[2-(dimethylamino)acetyl]-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(3-methoxyphenyl)methyl]-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-methoxybenzamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
2-({4-cyclopropyl-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
3-({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-2,2-dimethylpropan-1-ol
1-benzyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine