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N-(4-chloro-2-fluorophenyl)-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}acetamide
2-({4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)phenol
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-methyl-1,3-thiazole-4-carboxamide
1-{4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
5-[(adamantan-1-ylmethyl)(methyl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[2-(2,3-dimethylphenoxy)ethyl]-4-(furan-2-carbonyl)-1,4-diazepane
N-[(3-methyl-1-benzofuran-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
benzyl N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)amine
(3aS,6aS)-5-[(4-fluoro-3-methoxyphenyl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1s,4s)-4-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]cyclohexan-1-amine
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
1-{4-[3-({[3-(trifluoromethyl)pyridin-2-yl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
(2R,3R,6R)-3-phenyl-5-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-methoxy-4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenol
4-{5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
1-(4-{[4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
(but-2-yn-1-yl)({[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl})(furan-2-ylmethyl)amine
ethyl 1-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)piperidine-2-carboxylate
5-{[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-cyclobutaneamido-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylbenzamide
3-phenyl-N-[1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
4,6-dimethyl-1-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
methyl 2-[bis(prop-2-en-1-yl)sulfamoyl]-6-{[4-(dimethylamino)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
({5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-(2-methylphenyl)-1,4-diazepane
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
4-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N,N-diethyl-1-{[4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-3-carboxamide
(3S,4R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-methylpiperidine-3,4-diol
(1S,5R)-6-(3-chlorobenzoyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aS)-5-[(3,4-dimethoxyphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1R,3S,5S)-8-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-8-azabicyclo[3.2.1]octan-3-ol
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2,3-difluorophenyl)acetamide
2-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]pyrimidine
9-methoxy-7-(5-methylthiophen-2-yl)-4-(pyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
ethyl 1-[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]piperidine-4-carboxylate
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
7-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-chloro-4-({1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide