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N,N-diethyl-2-(6-methoxynaphthalen-2-yl)morpholine-4-carboxamide
1-({1-[(1-ethylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)piperidine-3-carboxamide
4-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine-4-carbonyl}morpholine
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol
2-[4-chloro-2-({2-oxo-1,3-dioxa-8-azaspiro[4.5]decan-8-yl}methyl)phenoxy]acetic acid
6-(morpholin-4-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
3-[5-(cyclopent-3-en-1-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
(2S,4R)-4-amino-N-[2-(1H-indol-3-yl)ethyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methoxypropan-1-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-hydroxyethyl)acetamide
2-(2-methoxyphenyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine
1'-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-methyl-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
1-[2-(3-chlorophenyl)ethyl]-4-{[(6-methylpyridin-2-yl)methyl]amino}pyrrolidin-2-one
1-{1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}piperidin-3-ol
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5,6,7,8-tetrahydroquinolin-2-yl)pyrrolidin-3-yl]methanol
(3S,4S)-1-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-4-propylpyrrolidine-3-carboxylic acid
4-cyclobutanecarbonyl-2-(3-phenylpropyl)morpholine
[5-({methyl[2-(2-methylpiperidin-1-yl)ethyl]amino}methyl)furan-2-yl]methanol
2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-N-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
5-(2,2-dimethyloxan-4-yl)-4-phenyl-1H-imidazole
N-{4-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]phenyl}acetamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-(3-hydroxyphenyl)acetamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-2-(morpholin-3-yl)acetamide
1-benzyl-5-[(4-methoxyphenyl)methyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{[4-(6-oxo-1,6-dihydropyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
1-(3-chlorophenyl)-4-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine
5-[6-amino-5-cyano-4-(2-methoxypyrimidin-5-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
N-(butan-2-yl)-N-(pyridin-3-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
1-[2-(dimethylamino)-4-({1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}acetamide
1-cyclopentyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide
6-(2-hydroxyethyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(phenylamino)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-5-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-{2-[(4-methyl-1H-imidazol-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
1-[2-(oxolan-2-ylmethoxy)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{1-[(2-methylphenyl)methyl]-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
7-methoxy-1-methyl-N-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-methyl-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
methyl 1-[2-hydroxy-3-(3-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
(3aS,6aS)-2-ethyl-1-oxo-5-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,7aR)-1-[(3,4-dimethylphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 5-(2,2-dimethylpropanoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{5-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-cyclopropyl-9-[2-(2-hydroxyethoxy)ethyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
ethyl 5-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[4-({8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)phenyl]acetamide