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1-(3-methoxybenzoyl)-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine
1-[(4aS,8aS)-4a-hydroxy-7-(1H-imidazol-2-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-cyclopentylethan-1-one
1-(pyridin-2-yl)-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethan-1-ol
N-[(2-methylphenyl)methyl]-3-(1-methylpiperidin-3-yl)-N-(prop-2-en-1-yl)propanamide
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[2-methoxy-5-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methoxypyridine-3-carbonitrile
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2,3,6-trifluorophenyl)acetamide
1-(4-fluoro-3-methoxyphenyl)-2-(furan-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
3-(1H-pyrazol-1-ylmethyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
3-(4-{[4-(6-oxo-4-propyl-1,6-dihydropyrimidin-2-yl)phenyl]methyl}piperazin-1-yl)propanamide
N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-({[(2-phenyl-1,3-oxazol-4-yl)methyl]amino}methyl)pyrrolidin-3-ol
4-(2H-1,3-benzodioxol-5-yl)-1-{2-[2-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(2-phenylquinoline-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(2-fluoro-4-methylbenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-[(3,4-dimethoxyphenyl)methyl]-2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-(2-methanesulfonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-(trifluoromethyl)benzamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-ethyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 1-{2-hydroxy-3-[4-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
4-({1-[3-(furan-2-yl)phenyl]piperidin-4-yl}amino)butan-1-ol
5-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
4-(3-ethylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(4-hydroxyphenyl)methyl]piperidine-3-carboxamide
N-{2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}methanesulfonamide
1-(4-benzylpiperazin-1-yl)-3-[1-(thiophene-3-carbonyl)piperidin-3-yl]propan-1-one
2-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,2,3,4-tetrahydroisoquinoline
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-methoxy-2,2-dimethylpropan-1-one
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-(5-phenyl-1H-pyrazole-3-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
3-(benzenesulfonyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)propanamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
2-(3-{3-[2-(trifluoromethyl)phenyl]phenyl}-1H-pyrazol-1-yl)acetamide
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
1-(difluoromethyl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
5-propyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[(2,4-dimethoxyphenyl)methyl]-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
1-[(4aR,8aR)-4a-hydroxy-7-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-(4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
8-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]quinoline
2-methoxyethyl 3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-(3-phenylpropyl)piperidin-4-amine
[(3R,5R)-1-(5-methoxypyrimidin-2-yl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
2-(3,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
(3-{2-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
4-(4-methyl-1H-pyrazol-1-yl)-1-(pyrrolidine-1-sulfonyl)piperidine-4-carboxylic acid
1-(4,7-dimethylquinazolin-2-yl)-N-(1-methoxypropan-2-yl)azepan-4-amine