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2-[5-(dimethyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
N-{1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxopentan-2-yl}acetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)methanesulfonamide
5-benzenesulfonamido-1-ethyl-2-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4-diazepane
9-methoxy-N-methyl-7-oxo-3-(quinolin-6-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,2,3-benzotriazole-5-carboxamide
3-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-propylpyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(cyclopropylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methyl-1,3-thiazole-5-carboxamide
6-(2-aminoethyl)-2-(3-methoxyphenoxymethyl)-3,4-dihydropyrimidin-4-one
(3R,4R)-1-(4-ethylbenzenesulfonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
methyl 5-({2-chloro-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(1S,5R)-3-benzyl-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 1-benzyl-3-cyclopropaneamido-5-({[3-(2-hydroxyethoxy)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-{[(4-chlorophenyl)methyl]sulfanyl}ethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 4-benzyl-1-[(3-chloro-4-hydroxyphenyl)methyl]piperidine-4-carboxylate
2-{2-[4-(oxolane-2-carbonyl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
2-[2-(4-chlorophenyl)morpholin-4-yl]-N,N-dimethylpyridine-3-carboxamide
methyl 5-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-{6-[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
N-({7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2S)-1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-methyl-2-(pyridin-3-yl)quinoline
1-(dimethylsulfamoyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(propan-2-yl)acetamide
(1R,2R)-2-phenyl-N-propyl-N-(pyridin-3-ylmethyl)cyclopropane-1-carboxamide
(3S,4R)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-N,N-dimethyl-6-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(4-chlorophenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}butanamide
4-methoxy-3-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-[(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
2-[3-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)phenoxy]acetamide
1-(2,3-dimethoxybenzoyl)-3-propylpiperidine-3-carboxylic acid
1-(2-chlorophenyl)-3-{1-[1-(2-ethylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{[4-(6-methoxypyridin-3-yl)phenyl]sulfanyl}acetamide
2-tert-butyl-6-(2-chloro-6-fluorobenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-2-ylsulfanyl)propanamide
N-(furan-2-ylmethyl)-4-[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]pyridine-2-carboxamide
N-{1-[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
1-{1'-[(6-methylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
1,3-dimethyl-6-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,1-dimethylazepane-2-carboxamide
1-{2-[5-(2-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-1H-1,2,3-triazole