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1-[1-(2-fluorophenyl)piperidin-4-yl]-3-(1-methyl-1H-1,3-benzodiazol-5-yl)urea
(4aR,8aS)-1-(2-cyclohexylethyl)-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
1-(2-methoxyethyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]piperidine-4-carboxamide
(3aR,6aR)-2-[6-(morpholin-4-yl)pyrimidin-4-yl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-2,6-dimethylpyridine-4-carboxamide
(1R,3S)-7-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-7-azaspiro[3.5]nonane-1,3-diol
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(4-fluoro-2-methoxyphenyl)methyl]amine
5-fluoro-N4-methyl-N2-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrimidine-2,4-diamine
methyl 4-[2-amino-3-cyano-6-(2-methylpropanoyl)-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl]-1H-pyrazole-3-carboxylate
N-{4-fluoro-3-[({2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}carbamoyl)amino]phenyl}propanamide
3-methyl-N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]thiophene-2-carboxamide
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]propanamide
N-methyl-4-(piperidin-3-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
9-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-6-oxa-9-azaspiro[4.5]decane
methyl 4-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
methyl 8-[3-(furan-2-yl)-3-phenylpropanoyl]-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N3-tert-butyl-1-cyclohexyl-N5-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)morpholine-2-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
4-chloro-5-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-4-hydroxy-2-(pyridin-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
(4aR,8aR)-4-[(8-methylquinolin-5-yl)methyl]-octahydro-2H-1,4-benzoxazine
N-cyclopropyl-2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
[2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-1,3-thiazol-4-yl]methanol
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
1-{4-[(2-hydroxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(thiophen-2-yl)ethan-1-one
8-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,8aS)-2-[(5-methyl-1H-indol-3-yl)methyl]-decahydroisoquinolin-4a-ol
4-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]benzoic acid
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,6-dimethoxy-N-(5-oxo-1-phenylpyrrolidin-3-yl)pyridine-3-carboxamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-methanesulfonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
1-({5-[(3,4-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
7-methyl-3-[(3-oxo-1,4-diazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
2-(4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}-6-methylpyrimidin-2-yl)phenol
5-(2,2-dimethyloxan-4-yl)-1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 2-oxo-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-benzyl-4-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-1,4-diazepan-6-ol
2-methoxy-N-[1-(2-phenylethyl)-7-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-5-yl]acetamide
1-cyclopentyl-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-6-oxopiperidine-3-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]propanamide