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N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-propanoylpiperidine-3-carboxamide
1-(4-{3-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2,2-dimethyloxan-4-yl)-1H-pyrazole-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxy-2-methylpropan-1-one
4-{2-methoxy-4-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}-1-methylpiperidine
3-(2-{1-methyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)pyridine
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
6-ethoxy-3-[(2-methylpiperidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
1-(4-{2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
1-[5-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-{[4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
2-(6-aminopyridin-3-yl)-2-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetic acid
4-(3-hydroxy-3-methylbutyl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]benzamide
[(3R,4R)-1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-oxo-1-phenyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]pyrrolidine-3-carboxamide
3-(propan-2-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,2-oxazole-5-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
1-(6-hydroxy-4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-(5-ethyl-1,3-oxazole-4-carbonyl)piperazin-2-one
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-propyl-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
5-(2-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1H-1,2,4-triazole
5-methyl-2-(3-methylthiophen-2-yl)-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-butanamido-N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-N-methylbenzamide
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3-carboxamide
[(2-chloropyridin-3-yl)methyl](methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-[1-(2,2-dimethylpropyl)-4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-cyclopentyl-N-[3-(1H-indol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
5-fluoro-N4,N4-dimethyl-N2-[(5-methylpyrazin-2-yl)methyl]pyrimidine-2,4-diamine
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidine
1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
2-methyl-6-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]-3,4-dihydropyrimidin-4-one
N-[(1-methylpiperidin-3-yl)methyl]-5-phenoxyfuran-2-carboxamide
8-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(furan-2-yl)-2-[5-methyl-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N,N-dimethyl-3-[(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
2-[4-(1-benzofuran-2-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
1-[1-(2-methoxyphenyl)propan-2-yl]-1-methyl-3-(6-methylpyridin-3-yl)urea
2-ethyl-7-{[2-(furan-2-yl)azepan-1-yl]methyl}-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
N-(1-benzothiophen-2-ylmethyl)-5-(2,4-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3,5-dimethyl-1-(propan-2-yl)-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
(4S)-1-(2,6-difluoro-3-methoxybenzoyl)-3,3,4-trimethylpiperidin-4-ol
(3S,4S)-1-[(4-methanesulfonylphenyl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
1-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-ethyl-4-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
2-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylpyridine-3-carboxamide