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3-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-2-yl]pyridine
N,5-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(1,3-thiazol-2-yl)piperazine
6-(2,2-dimethylmorpholin-4-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
6-tert-butyl-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-indole-6-carboxamide
(3R,7S,8aS)-3-(2-methylpropyl)-7-({[3-(methylsulfanyl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3,3-dimethyl-1-{[5-(piperidin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
(3S,4R)-1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
6-methyl-4-oxo-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-N,N-bis(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1-{2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetyl}piperidine-4-carboxamide
(3R,9R)-11-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-phenyl-N-propylimidazo[1,2-a]pyridine-6-carboxamide
methyl (2S,4R)-1-methyl-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-amido}pyrrolidine-2-carboxylate
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-oxo-2-phenylacetamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(trifluoromethyl)benzamide
ethyl 4-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidine-1-carboxylate
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
3-methyl-7-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-hydroxy-N-(2-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}ethyl)acetamide
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N-methylpyrimidin-4-amine
2-(carbamoylamino)-N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-{3-acetamido-5-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}acetamide
4-({1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}methyl)morpholine
4-({4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
3-ethyl-N-(2-methoxyethyl)-4-methyl-N-propyl-1H-pyrazole-5-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1-[(1R)-1-phenylethyl]-1H-imidazole
5-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N,N-dimethylpyridin-2-amine
ethyl 1-(cyclopropylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-(3-chloro-4-methoxyphenyl)-N-[2-(5-methylfuran-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N4-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methylpyrimidine-2,4-diamine
(2R,3S,6R)-5-(5-chloropyridine-2-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
N-(1-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]-4-(pyridin-4-yl)piperidine-1-carboxamide
(4aS,7aR)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-cyclopropyl-2-{4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]morpholin-3-yl}acetamide
2-[2-(3-hydroxyadamantan-1-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-methyl-2-{4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]phenyl}propanenitrile
4-(4-cyclopentylpyrimidin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2-fluorophenyl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-pyrazole-5-carboxamide
2-(5-{5-[(methylsulfanyl)methyl]furan-2-yl}-3-phenyl-1H-1,2,4-triazol-1-yl)acetic acid
2-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
(2S,4S)-4-amino-1-[3-(N-methylmethanesulfonamido)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,4R)-3-cyclobutyl-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-methylpyrrolidin-3-ol
2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}acetamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-hydroxy-3-methylbenzamide