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4-({3-[(dimethylamino)methyl]-4-hydroxyphenyl}methyl)-1-(3,5-dimethylphenyl)piperazin-2-one
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](furan-2-ylmethyl)amino}butan-1-ol
5-(benzylamino)-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-4-phenylbenzamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{[methyl(2-methylpropyl)amino]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
methyl N-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}carbamate
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-[2-(4-hydroxyphenyl)acetyl]pyrrolidine-2-carboxamide
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-chloro-4-(cyclopropylmethyl)-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
ethyl 1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
6-ethyl-N4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methylpyrimidine-2,4-diamine
2-(2-{methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(4aR,7aS)-1-cyclopropanecarbonyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,5R)-1-(3-chloro-1H-indole-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-[(1-benzylpyrrolidin-3-yl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
3-(1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}piperidin-3-yl)benzoic acid
2-(5-fluoro-2-methoxyphenyl)-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
9-ethyl-1-methyl-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4R)-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
2-{[4-(6-methylpyridazin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
3-(2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamido)propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
methyl[1-(pyrazin-2-yl)propan-2-yl]{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
2-[4-(3-fluoropyridin-2-yl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
4-(1-cyclohexyl-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1H-1,2,4-triazol-3-yl)pyridine
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N,N-diethylacetamide
(4aS,8aR)-6-(2,4-dimethylpyrimidine-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
9-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3-oxa-9-azaspiro[5.5]undecane
2-{[1-(dimethyl-1,3-thiazol-2-yl)propyl]amino}propane-1,3-diol
2-(1H-1,3-benzodiazol-1-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})(quinoxalin-5-ylmethyl)amine
(1S,5R)-3-(pyridin-3-ylmethyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[1-(4-methylpentanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(3-{[1-(1-benzyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}acetamide
4-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
(4aS,7aR)-N-(3-chloro-4-methoxyphenyl)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[N-methyl3-(3-cyanopiperidine-1-carbonyl)benzenesulfonamido]propanamide