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N-methyl-2-(3-oxo-1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperazin-2-yl)acetamide
3-[5-(6-methylpyridazin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[2-(piperazin-1-yl)ethyl]benzamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}cyclohex-3-ene-1-carboxamide
(2S)-1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-2-(pyrrolidin-1-ylmethyl)pyrrolidine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(oxan-4-yl)piperidin-3-ol
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-phenylpiperazine
[(4-chlorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-phenyl-N-[(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
1-(2-phenylethyl)-3-(propan-2-yl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}acetamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2-fluorophenyl)methyl]piperidine
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}but-2-ynamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
N-[2-(1H-pyrazol-1-yl)ethyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(2-ethoxyphenyl)methyl]piperidine
ethyl 4-[1-(3-chlorobenzoyl)piperidin-3-yl]piperazine-1-carboxylate
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-2-(2-oxopiperidin-1-yl)acetamide
4-cyclopentanecarbonyl-1-(2-methylphenyl)piperazin-2-one
1-(4-{2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
5-[1-(2-fluorophenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
2-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)quinoline
6-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrazine-2-carboxamide
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-3-(2-ethoxyethyl)-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-chloro-1-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[2-(3-acetamidopropanamido)-4-methylphenyl]-2-methylbenzamide
2-amino-3-ethyl-N-[(4-sulfamoylphenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(methoxymethyl)-5-(1-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-1H-imidazol-2-yl)pyrimidine
(1R,3S)-7-(2-chloro-6-fluoro-3-methylbenzoyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-phenylpentanamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(pyrimidin-4-ylmethyl)benzamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-[(4-methylpiperidin-1-yl)methyl]furan-2-carboxamide
N-(2-methoxy-2-methylpropyl)-3-{[(1-methylpiperidin-2-yl)methyl]sulfamoyl}benzamide
N-methyl-3-(piperidin-3-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
1-(pyridin-3-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(4aS,8aR)-1-(2-aminoethyl)-6-(1H-indole-6-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-({1-[6-(4-fluorophenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-(1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-1H-1,3-benzodiazole
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(6-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-(4-methoxy-2-methylphenyl)-3-[1-(quinoline-3-carbonyl)piperidin-3-yl]propanamide
2-methyl-8-[6-(propan-2-yl)-1H-indole-2-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)-5-[(furan-2-ylformamido)methyl]benzoate
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-[(2S)-2-(methylamino)propanoyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-{3-[3-(5-fluoropyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
4-(6-aminopyridin-3-yl)-2,2-diphenylbutanenitrile
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-imidazol-2-yl]-1-ethyl-1H-1,2,4-triazole