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1-[benzyl(methyl)amino]-3-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-hydroxy-4-methoxy-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]benzamide
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(3-methylpyridin-2-yl)methyl]acetamide
3-{[(1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-(phenylsulfanyl)ethan-1-one
4-[(3-methoxypropyl)amino]-5-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
2-{3-methyl-5-phenyl-[1,2]thiazolo[5,4-b]pyridin-6-yl}-1H-imidazole
1-{4-[(quinolin-8-yl)amino]piperidin-1-yl}ethan-1-one
3-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)propan-1-ol
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
4-(4-{[2-(4-methoxyphenyl)ethyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
N1-[4-(4-chlorophenoxy)phenyl]-N3-methylpiperidine-1,3-dicarboxamide
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]-N-(4-methylphenyl)-3-oxopropanamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[3-(propan-2-yloxy)propyl]acetamide
1-(4-{2-methoxy-5-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
2-(2-methoxyethyl)-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(4-methyl-1H-pyrazol-1-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine-4-carboxylic acid
(1R,5R)-N-[2-(methylsulfanyl)phenyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N,N-dimethyl-3-[(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}-N-propylpiperidine-1-carboxamide
4-[5-methyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
N-(2,2-diphenylpropyl)oxane-2-carboxamide
3-{2-[4-(1H-pyrazol-3-yl)benzoyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
5-(2-methylpentanoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-4-methylphenol
(2S,4S,5R)-5-(2-fluorophenyl)-4-[(3-hydroxypropyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyridin-3-ol
1-methyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrrole
4-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)morpholine
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-amine
methyl 1-ethyl-3-(oxolane-3-amido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-3-[N-methyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
2,2-dimethyl-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)propanamide
N-[1-(6-methylpyridin-2-yl)propan-2-yl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
3-[(cyclohexylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
5-cyclopropyl-N-(2-hydroxybutyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-[(6-methylpyridin-3-yl)oxy]-1-(oxane-2-carbonyl)piperidine-4-carboxylic acid
2-(ethylamino)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
1-(morpholin-4-yl)-2-[4-({[2-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)phenoxy]ethan-1-one
ethyl N-{[(2S,4S)-1-[(4-chlorophenyl)methanesulfonyl]-4-fluoropyrrolidin-2-yl]methyl}carbamate
(1R,3S)-3-methoxy-7-(3-phenoxybenzoyl)-7-azaspiro[3.5]nonan-1-ol
methyl 6-[2-(4-fluorophenyl)acetyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2H-1,3-benzodioxol-5-yl)-2-(acetamidomethyl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-N-(3-chloro-4-methylphenyl)piperidine-1-carboxamide
3-[4-(dimethylamino)phenyl]-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]propanamide