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4-[1-(thiophene-2-sulfonyl)piperidin-3-yl]morpholine
3-(5,6-dimethylpyridin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
2-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(2S)-3-phenyl-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}propan-1-ol
2-({[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl](methyl)amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-({2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-2,6-dimethylphenyl acetate
1-(4-phenylbenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(1s,4s)-4-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-ol
2-[(pyridin-2-ylmethyl)(quinoxalin-2-ylmethyl)amino]butan-1-ol
3-(5-methylthiophen-2-yl)-N-(propan-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(1-cyclopentanecarbonylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-3-carboxamide
N1,N1,N4-trimethyl-N4-[(1-phenylpyrrolidin-3-yl)methyl]piperidine-1,4-dicarboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-[(2-methoxyphenyl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-phenyl-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(2,4-dichlorophenoxy)acetamide
3-{2-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
5-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)-N-(4-methoxyphenyl)-1,3-thiazol-2-amine
N-butyl-3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
6-methoxy-N-methyl-N-[(3-methylpyridin-4-yl)methyl]pyrimidin-4-amine
2-(3-{3-[2-(dimethylamino)-6-methylpyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)-N-(propan-2-yl)acetamide
1-cyclopropanecarbonyl-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidine
2-amino-4-ethyl-N-methyl-N-(quinoxalin-2-ylmethyl)-1,3-thiazole-5-carboxamide
1-cyclobutanecarbonyl-N-methyl-N-(quinolin-6-ylmethyl)piperidine-4-carboxamide
1-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide
N-(2-fluoro-4-methylphenyl)-4-(4-methoxybutyl)piperazine-1-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
3-ethyl-4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
2-(2-methoxyphenyl)-8-methyl-5-(quinoxalin-6-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-chloro-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]pyridine-4-carboxamide
2-(3-fluorophenyl)-1-[3-(2-phenylacetyl)piperidin-1-yl]ethan-1-one
3-[4-(hydroxymethyl)phenyl]-N-(propan-2-yl)benzamide
N-methyl-N-(1-{1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
8-benzyl-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridin-2-ol
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(quinoxaline-5-carbonyl)-1,4-diazepan-2-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
5-[2-(3-methoxyphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-(1-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)carbamoyl]methyl}-1H-pyrazol-4-yl)furan-2-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyridin-3-ol
1-(2-cyclohexylethyl)-3-hydroxy-3-({3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)piperidin-2-one