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N-[3-(1H-imidazol-1-yl)propyl]-2-(trifluoromethyl)pyrimidin-4-amine
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
2-(3,4-dichlorophenyl)-4-[5-(propan-2-yl)pyrimidin-4-yl]morpholine
(2S,4S)-1-[(4-methoxy-3-methylphenyl)methyl]-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(quinolin-4-ylmethyl)amine
2-[2-(dimethylamino)ethyl]-9-[2-(methylamino)pyrimidine-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-{[4-(2-fluorophenyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
N-({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
2-phenyl-5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidine
2,6-dimethyl-4-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
7-(1-benzothiophen-3-yl)-4-[5-(methoxymethyl)furan-2-carbonyl]-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(butan-2-yl)({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
[(3R,5S)-5-(hydroxymethyl)-1-[(4-phenylphenyl)methyl]piperidin-3-yl]methanol
2-amino-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperidine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
2-[(4-methylphenyl)sulfanyl]-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
methyl[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl](4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
5-butyl-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}pyridine
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-(furan-3-carbonyl)piperidine
1-({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperidine-4-carbonitrile
5-(pyrrolidin-1-yl)-2-(pyrrolidin-3-ylmethyl)-2,3-dihydropyridazin-3-one
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(diethylamino)ethan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-1-methylazepane-2-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
2-hydroxy-5-{1-[2-methyl-2-(morpholin-4-yl)propyl]-1H-imidazol-2-yl}benzoic acid
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-fluorophenyl)methyl]piperidine
5-[3-(methylsulfanyl)propyl]-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3S,4S)-4-(piperidin-1-yl)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-ol
5-(2-chloroprop-2-en-1-yl)-7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-{1-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
ethyl 4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidine-1-carboxylate
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-{3-[4-({[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}amino)piperidin-1-yl]phenyl}cyclopropanecarboxamide
2-[3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenoxy]acetamide
(3S,4R)-1-[2-(pyridin-3-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-[5-(3-cyclopropyl-1H-pyrazol-4-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]pyridine
2-(4-methyl-1,3-oxazole-5-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl})methylamine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
2-(4-chlorophenyl)-4-(5-ethyl-1,3-oxazole-4-carbonyl)morpholine
3-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonan-9-ol
N-[(2R,4S,6S)-2-(3,5-difluorophenyl)-6-[(E)-2-phenylethenyl]oxan-4-yl]acetamide
5-{[2-(benzylamino)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1,4-dioxan-2-ylmethyl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
(1S,4S)-2-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane