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2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2,4-dichlorophenoxy)acetamide
2-[4-(dimethylamino)phenyl]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(benzyloxy)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
4-[(3,4-dimethoxyphenyl)methyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
6-[(3-phenoxyazetidin-1-yl)methyl]pyridine-2-carboxylic acid
2-(3-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
[5-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)furan-2-yl]methanol
[(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
3-[(3S,4R)-1-benzyl-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
1-[2-(1-benzofuran-2-yl)phenyl]piperazine
4-(2-chloro-6-fluorobenzoyl)-1-(4-methylphenyl)piperazin-2-one
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-ethylpiperazin-2-one
2-ethyl-4-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1-methylcyclopropanecarbonyl)piperidin-3-yl]propanamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(2,5-dimethylphenyl)ethyl]-3-propanamidobenzamide
1-(azocan-1-yl)-3-[5-methoxy-2-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-cyclopentyl-3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-5-(phenylsulfamoyl)benzamide
2-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]-N-(5-fluoro-2-methylphenyl)acetamide
5,6-dimethoxy-2-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-1,2-dihydroisoquinolin-1-one
2-(3-methyl-1H-pyrazol-1-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-[3-(propan-2-yl)-5-[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]-1H-1,2,4-triazol-1-yl]pyridine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-(oxolan-3-yl)-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazole
1'-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}spiro[indene-1,4'-piperidine]
(1S,4S)-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(1-methanesulfonylpiperidin-4-yl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
4-[(3-fluorophenyl)methyl]-11-[4-(pyridin-2-yl)piperazin-1-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-3-(3-fluorophenoxymethyl)piperidine
N-(furan-2-ylmethyl)-2-(pyridin-3-yl)-N-(thiophen-2-ylmethyl)pyrimidine-5-carboxamide
1-(1-ethyl-6-oxopiperidine-3-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-[4-(4-cyclohexylpiperazine-1-carbonyl)piperidin-1-yl]-2-[(3,4-dimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(9H-purin-6-yl)quinoline
4-[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-3-(3-methoxyphenyl)propan-1-one
N-[(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[(4-methylphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazin-2-one
4-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-{2-[2-(trifluoromethyl)phenyl]ethyl}oxolane-3-carboxamide
(3R,5S)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
1-[2-methoxy-5-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N5-cyclooctyl-1-(2-methoxyethyl)-N3-methyl-4-oxo-N3-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide