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4-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenol
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
4-methoxy-6-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[3-(oxolan-3-yl)propyl]amine
(5S,9aS,9bS)-5-(3-ethoxyphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2R)-1-hydroxybutan-2-yl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
4-(5-{2-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyridin-4-ylsulfanyl)acetamide
5-cyclobutanecarbonyl-3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[4-({4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
3-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
ethyl 2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]acetate
N-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-2-carboxamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
1-(2-methoxyacetyl)-N,4-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazine-2-carboxamide
5-(1-benzofuran-2-yl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1,2,4-triazin-3-amine
N-methyl-4-sulfamoyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
11-(4-acetylpiperazin-1-yl)-4-[(2-chlorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{[3-(5-fluoro-4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}-N,N-dimethylpiperazine-1-carboxamide
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(3-methylphenyl)methyl]amine
N-[1-(methoxymethyl)cyclopentyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-benzyl-N-methyl-3-({[2-(4-methyl-1H-imidazol-2-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(1H-imidazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
1-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]cyclopropan-1-amine
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(pyrimidin-5-yl)-1H-pyrazol-1-yl]acetamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-(4-methanesulfonyl-1,4-diazepan-1-yl)propan-1-one
3-methyl-2-[1-(oxan-3-yl)-4-phenyl-1H-imidazol-5-yl]-1H-indole
3-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-propyl-1-benzofuran-2-carboxamide
3-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,2-dihydroquinoxalin-2-one
(2S,4S)-4-amino-N-ethyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidine-2-carboxamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methylpyridazin-3-amine
N-cyclopropyl-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2H-chromene-3-carboxamide
1-cyclopentanecarbonyl-N-{3-[(pyridin-3-yl)amino]propyl}piperidine-4-carboxamide
1,9-dimethyl-4-[2-(pyridin-3-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1H-imidazol-2-ylmethyl)piperidine-3-carboxylate
1-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(1,1-dioxo-1λ6-thiolan-3-yl)urea
9-hydroxy-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-[1-(6-chloroquinolin-4-yl)piperidin-4-yl]piperidin-3-ol
4-benzyl-3-(1-butanoylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]pyrimidin-4-yl}amino)acetic acid
2-(4-acetylphenoxy)-N-(1,4-dioxan-2-ylmethyl)acetamide
8-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 6-butanoyl-2-[(4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(3-fluorophenyl)propanoyl]piperidin-3-yl}propanamide
N-ethyl-2-[4-(2-phenoxyacetyl)piperazin-1-yl]pyridine-3-carboxamide
2-(2-chlorophenyl)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[4-(ethanesulfonyl)piperazin-1-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
2-(3,4-dichlorophenyl)-4-[(2-methoxypyrimidin-5-yl)methyl]morpholine
4-({4-[(3-methoxypropyl)amino]-6-methylquinazolin-2-yl}methyl)piperazine-1-carbaldehyde