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4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
{2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-4-yl}methanol
N-(1H-indol-2-ylmethyl)-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(methylamino)pyrimidin-2-yl]-decahydro-1,6-naphthyridin-2-one
3-ethyl-1-methyl-4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
3-[({3-azaspiro[5.5]undecan-9-yl}amino)methyl]-1λ6-thiolane-1,1-dione
4-[(4-fluoro-3-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-[cyclopropyl(4-methoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-({1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]piperidin-3-yl}methyl)pyrrolidin-2-one
4-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1-methylpiperazin-2-one
1-(1-benzofuran-3-carbonyl)-2-(thiophen-2-yl)azetidine
1'-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-amino-6-(furan-2-yl)-4-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
(2S,4R)-N-cycloheptyl-1-[(4-ethylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
5-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-N,N-dimethylfuran-2-carboxamide
1-[4-({3-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
2-(5-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
1-ethyl-4-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
1-cyclopropyl-4-({[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]amino}methyl)pyrrolidin-2-one
(4aR,7aS)-1-(2-methylpropanoyl)-4-[(2E)-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-chloro-N-(4-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)benzamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
1-tert-butyl-3-methyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-(3-hydroxy-3-methylbutyl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
7-fluoro-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-methyl-1H-indole-2-carboxamide
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[3-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(1H-imidazol-4-yl)-1-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1H-imidazole
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1-methylpiperidine-3-carboxamide
2-{9-[(3-fluorophenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
3-(1,2-oxazinan-2-yl)-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-1-one
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
5-ethyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,3-oxazole-4-carboxamide
3-methoxy-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
1-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-4-yl}piperidin-4-ol
4-({[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
2-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)-1,3-thiazole-4-carboxamide
1'-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[2-(dimethylamino)ethyl]-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-oxopyrrolidine-3-carboxamide
3-(hydroxymethyl)-1-(7-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-ol
ethyl 4-{4-[5-(oxolane-3-amido)-1H-pyrazol-1-yl]piperidin-1-yl}piperidine-1-carboxylate
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-(thian-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
7-[(3-methylphenyl)methyl]-2-(quinoline-6-carbonyl)-2,7-diazaspiro[4.5]decane
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}acetamide