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1-(4-{2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)ethan-1-ol
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(2-methoxypyridin-3-yl)pyridine-3-carbonitrile
(3S,4S)-4-(naphthalen-2-yl)-1-(pyridine-4-carbonyl)piperidin-3-ol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-phenylazepane
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-6-methylpyridine-3-carboxamide
N-[2-(2,5-dimethylphenoxy)ethyl]-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
1-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine-4-carbonitrile
(4aS,7aR)-1-[(4-acetylphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1H-imidazole-5-carboxamide
2-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[3-(pyridin-3-yloxy)propyl]acetamide
1-[1-(4-fluorophenyl)ethyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
[3-benzyl-1-(8-methoxyquinolin-2-yl)piperidin-3-yl]methanol
(4aS,7aR)-1-(1-methyl-1H-pyrazole-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
ethyl 5-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[2-methoxy-5-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(3R)-1-(2-methoxy-4,5-dimethylbenzenesulfonyl)-3,4,4-trimethylpyrrolidin-3-ol
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-(3-methoxypropyl)-4-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]piperazine
(5S,9aS,9bS)-5-(2-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-benzyl-1-[4-(1H-imidazol-1-yl)benzoyl]-N-methylpiperidin-3-amine
(2S,4R)-1-[2-(5-acetylthiophen-3-yl)acetyl]-4-amino-N-ethylpyrrolidine-2-carboxamide
2-hydroxy-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-2-hydroxy-5-methylbenzamide
2-(4-methanesulfonylphenyl)pyridine-4-carboxamide
N-[2-(2-fluorophenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-methyl-1'-[4-(1H-pyrazol-1-yl)butanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyrrolidine-1-carbonyl)piperidine
N-ethyl-2-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]pyridine-4-carboxamide
4-cyano-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
1-ethyl-4-({8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decan-1-yl}methyl)-1H-pyrrole-2-carbonitrile
2-(3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
1-methyl-6-(propan-2-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
8-{[3-(3-cyclohexylpyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}quinoline
5-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
N-{3-[2-(2-fluoro-4-methylphenyl)-1H-imidazol-1-yl]-4-methoxyphenyl}acetamide
methyl 2-chloro-5-({2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}amino)benzoate
2-(5-methyl-2-phenylfuran-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one