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2-ethyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
3,5-dimethyl-4-({[1-(morpholin-4-yl)cycloheptyl]methyl}carbamoyl)-1H-pyrrole-2-carboxylic acid
2-{3-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
3-[(furan-2-ylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
4-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
2-(3-methoxyphenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,3-oxazole-4-carboxamide
2-{imidazo[1,2-a]pyridin-3-yl}-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}acetamide
N-[2-(4-hydroxypiperidin-1-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
2-(methoxymethyl)-1-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-yl}-5-(trifluoromethyl)-1H-1,3-benzodiazole
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-one
{4-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]morpholin-2-yl}methanamine
2-{5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-(propan-2-yl)-3-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propanamide
N-methyl-N'-(4-methylphenyl)-N-(quinolin-2-ylmethyl)propanediamide
methyl 3-(2-chlorobenzenesulfonamido)-5-[(2-methylpropanamido)methyl]benzoate
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-benzyl-5-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)pyrimidin-2-amine
N-[1-(4-methanesulfonylphenyl)ethyl]-5,6-dimethylpyrimidin-4-amine
5-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-3-propylimidazolidine-2,4-dione
3-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-benzyl-5-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
ethyl 1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-(2,5-dimethylphenoxymethyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,2-oxazole-3-carboxamide
3-{2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
3-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-imidazol-5-yl}phenol
2-chloro-N-(propan-2-yl)-5-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]carbamoyl}amino)benzamide
N-(3-{4-[methyl(quinoxalin-6-ylmethyl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
7-(3-chlorophenyl)-4-(dimethyl-1,3-oxazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(1H-pyrazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[5-(aminomethyl)pyridin-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(thiophen-2-yl)acetamide
1-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]piperidin-4-ol
4-{[ethyl(oxan-4-ylmethyl)amino]methyl}-2,6-dimethylphenyl acetate
(2R,3R,6R)-3-(3-methoxyphenyl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(naphthalen-2-yloxy)-1-(thiophen-2-ylmethyl)piperidine-4-carboxylic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-3-yl]methanol
1-(furan-3-ylmethyl)-4-(2-phenylacetyl)-1,4-diazepane-6-carboxylic acid
N-(1-{7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[1-(4-fluorophenyl)piperidin-4-yl]acetamide
2-(4-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}quinazolin-2-yl)ethan-1-amine
2-[(3,4-difluorophenyl)methyl]-8-[2-(2-hydroxyethoxy)ethyl]-2,8-diazaspiro[4.5]decan-3-one
(2R,6R)-4-{5-[(dimethylamino)methyl]furan-2-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl 1-{2-hydroxy-3-[4-(piperidin-1-ylmethyl)phenoxy]propyl}piperidine-4-carboxylate
2-amino-4-[2-(2-methoxyethyl)pyrimidin-5-yl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(3aS,6aR)-5-{7-methylthieno[3,2-d]pyrimidin-4-yl}-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{2-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
5-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid