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1-(6-chloroquinolin-4-yl)-3-(hydroxymethyl)piperidin-3-ol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
7-(4-chlorophenyl)-2-(propoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-(cyclopropylmethyl)-2-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-[(4-fluoro-3-methoxyphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(2-methoxyphenyl)-3-{1-[1-(oxolane-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
4-[(4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}furan-2-yl)methyl]morpholine
1-[4-(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethan-1-one
ethyl 4-[(3S,4S)-4-hydroxy-1-(4-methoxybenzoyl)pyrrolidin-3-yl]piperazine-1-carboxylate
(1R,5S,6R)-3-[(2,2-dimethyloxan-4-yl)methyl]-N-(pyridin-3-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
[3-(2-methoxyethyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-3-yl]methanol
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylpropanamide
3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)pyrazolo[1,5-a]pyridine-2-carboxamide
1-(propan-2-yl)-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidin-2-one
1-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(prop-2-en-1-yl)urea
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(6-methylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
4-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-4-oxo-N-(1,3,4-thiadiazol-2-yl)butanamide
N-[1-({[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-4-fluorophenol
methyl 2-[({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]benzoate
8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-5-({4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)furan-2-carboxamide
1-{4-oxo-4-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]butyl}pyrrolidin-2-one
4-(3,3-diphenylpiperidine-1-carbonyl)-1-oxaspiro[4.4]nonan-2-one
(3E)-N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}pent-3-enamide
1-(2-methoxyethyl)-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-[(5-methylthiophen-2-yl)methyl]urea
5-fluoro-N,N-dimethyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-(4-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)imidazolidin-2-one
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
1-(3-{[(6-phenylpyridazin-3-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
(isoquinolin-5-ylmethyl)(methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
{4-[(4-fluoro-2-methylphenyl)methyl]-1-methylpiperazin-2-yl}methanol
N-(2-methoxyethyl)-1-methyl-N-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-amine
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2,2-diphenylethan-1-one
1-(2-methoxybenzoyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
2-oxo-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-dihydroquinoline-4-carboxamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(3-methyl-1H-indol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[1-(4-methylpentan-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-[(2R,3R)-1'-(3-ethynylbenzoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
4-(3,6-dimethylpyrazin-2-yl)-2-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenol
N-methyl-2-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrimidine-5-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine