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6-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-N-(pyridin-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(1,4-dimethyl-1H-pyrazol-5-yl)-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}benzamide
N-[2-(dimethylamino)ethyl]-N-ethyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
4-chloro-5-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
(1R,3S)-7-(4,4,4-trifluorobutyl)-7-azaspiro[3.5]nonane-1,3-diol
2-benzyl-4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-thiazole
4-[3-ethyl-5-(5-hydroxypyrazin-2-yl)-1H-1,2,4-triazol-1-yl]-1-methyl-1,2-dihydroquinolin-2-one
2-{[(4-ethoxypyrimidin-2-yl)amino]methyl}-6-methyl-3,4-dihydropyrimidin-4-one
N-{1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
(2R,3R)-1'-(6-methylpyridazin-3-yl)-3-(morpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-(1H-indol-1-ylmethyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1,2-dihydrophthalazin-1-one
4-{1-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]piperidin-3-yl}benzoic acid
2-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1H-1,3-benzodiazole
ethyl 5-[3-(2-chlorophenyl)propanoyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(3,4-dimethylphenyl)methyl]pyrimidin-2-amine
N-[(3-methoxyphenyl)methyl]-2-(pyrrolidin-3-yl)benzamide
5-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
methyl 3-[2-(naphthalen-1-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
3-[(1-cycloheptylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
4-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-6-methylpyrimidin-2-amine
2-{5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-indole
3-chloro-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
9-hydroxy-N-[1-(methylcarbamoyl)cyclohexyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(2-oxoimidazolidine-4-carbonyl)piperazin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
3-{[4-(diphenylmethyl)piperazin-1-yl]methyl}pyridin-2-amine
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-{[(naphthalen-1-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-amino-8-(1-cyclopentylpiperidine-3-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-amino-4-(1-ethyl-1H-pyrazol-4-yl)-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
2-{1-[(6-methylpyridin-2-yl)methyl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
(2R,3R,6R)-3-(3-methoxyphenyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)piperidin-2-one
ethyl 1-[3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3-carboxylate
5-(pyrrolidin-2-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}thiophene-2-carboxamide
N-cyclohexyl-2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methylacetamide
6-[(diethylamino)methyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(9H-purin-6-yl)-decahydroisoquinoline
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-(1,3-dihydro-2-benzofuran-5-yl)-3-[(2,2-dimethylpropyl)amino]-5-[(propan-2-yl)sulfamoyl]benzamide
5-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
7-(morpholin-4-ylmethyl)-4-(5-phenyl-1,2-oxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[(4-phenyloxan-4-yl)methyl]propanamide
9-(2-butoxyacetyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-methylpyrimidine-5-carboxamide