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N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-[1-(2H-1,3-benzodioxol-5-yl)-5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-1H-1,2,4-triazol-3-yl]acetamide
5-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
4-(2-methoxyethyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-(6-methoxy-2H-1,3-benzodioxol-5-yl)-3-[3-(4-methyl-1,3-thiazol-2-yl)propyl]urea
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(3-hydroxy-3-methylbutyl)(methyl)amino]methyl}piperidin-2-one
1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
1-(methoxymethyl)-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-propylpyrrolidin-3-yl]cyclobutane-1-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-3-methylphenyl)-1H-pyrazole
2-methyl-6-(piperidin-3-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidin-4-amine
6-oxo-N-(pyridin-4-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-(1,3-oxazole-5-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-methyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyridine-4-carboxylic acid
methyl 3-(4-cyanopiperidine-1-carbonyl)-5-(cyclobutylmethoxy)benzoate
3-({2-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(4-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3-ethoxypropyl)-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
3-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-2-methyl-1,3-benzothiazole
4-(1-ethyl-1H-pyrazole-4-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
8-(5-acetylpyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2S)-oxolan-2-ylmethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(3R,4R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-3-methyl-3-phenylpiperidine
2-cyclopropyl-1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-imidazole
7-methoxy-3-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-(3,4-dimethoxyphenyl)piperidin-3-amine
5-hydroxy-2-(4-methyl-3-phenylpiperazine-1-carbonyl)-4H-pyran-4-one
4-{5-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]pentyl}morpholine
1'-methyl-5-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-3,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(4-chlorophenyl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}thiophene-3-carboxamide
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](ethyl){[2-(prop-2-en-1-yloxy)phenyl]methyl}amine
2-[2-({[2-(dimethylamino)-2-(3-methylphenyl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide
1-(4-fluorophenyl)-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}butane-1,4-dione
N-[(1R,3R)-3-aminocyclopentyl]-2-oxo-2-phenylacetamide
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
2-(1,2-benzoxazol-3-yl)-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
N,3-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-(phenoxymethyl)furan-2-carboxamide
5-(4-acetyl-4-phenylpiperidine-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
1-(1,4-dithiepan-6-yl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-(2-chloro-4-fluorophenyl)pyridin-2-ol
13-(2,3-dimethyl-1H-indol-7-yl)-4-methyl-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
7-fluoro-2-methyl-N-{3-[(pyridin-3-yl)amino]propyl}quinoline-4-carboxamide