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2-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
2-acetamido-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
2-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}-4-methoxypyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-(2-methylbenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(3-chlorophenyl)-4-[4-(pyrrolidin-1-yl)benzoyl]piperazin-2-one
2-cyclohexyl-5-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}pyrimidine
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
5-[4-(ethoxycarbonyl)piperazin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(2-methyl-5-sulfamoylphenyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[2-(dimethylamino)ethyl]-6-oxo-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
methyl 3-(2-chlorobenzamido)-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-[4-(3-methoxypyrazin-2-yl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
1-(5-fluoro-1H-indole-2-carbonyl)-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
5-chloro-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-2-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}urea
1-tert-butyl-5-oxo-N-[1-(pyrazin-2-yl)piperidin-4-yl]pyrrolidine-3-carboxamide
2-{4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperazin-1-yl}pyrimidine
1-[2-(benzyloxy)ethyl]-1,4-diazepane-6-carboxylic acid
5-(2-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
N-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
4-hydroxy-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
6-(4-fluorophenyl)-2-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
5-{4-hydroxy-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
1-(2,4-difluorophenyl)-3-(oxan-4-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-(3-fluoro-4-methylphenyl)-2-{[(1-methanesulfonylpiperidin-3-yl)methyl]amino}acetamide
(4aS,7aR)-1-[(3-methylthiophen-2-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
1-(oxolan-2-ylmethyl)-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
1-[(4-methoxyphenyl)methyl]-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperazin-2-one
(1S,5R)-6-(3-methyl-1H-pyrazole-5-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methanesulfonyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
1-{4-[4-(azepane-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
1-({5-[(2-methoxy-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-[2-({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
2-methyl-4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}quinoline
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyridine-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]ethan-1-amine
4-[(2-hydroxyethyl)sulfamoyl]-N-[2-(1H-pyrrol-1-yl)ethyl]benzamide
4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
ethyl 4-{1-[2-(2-chlorophenyl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
8-[(3-ethenylphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane
(2S,4R)-4-{4-[(1-adamantan-1-yl-N-methylformamido)methyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
2-(4-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]pyrimidine-5-carboxylic acid
3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one