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(1S,6R)-3-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
8-{[4-(difluoromethoxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aS,7aR)-1-(2-fluorobenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[(2S)-1-acetylpyrrolidine-2-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
2-[1-methyl-4-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperazin-2-yl]ethan-1-ol
2-[(2,6-dichlorophenyl)methyl]-N-ethyl-4-hydroxy-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(oxolane-2-carbonyl)piperazine
6-cyano-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
3-[3-({[2-(4-methoxyphenyl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-[(5-{[(1s,4s)-4-aminocyclohexyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]methanesulfonamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
4-(2,4-dimethylpyrimidine-5-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
2-{1-[(4-methanesulfonylphenyl)methyl]piperidine-3-carbonyl}pyridine
3-methyl-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
5-{1-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-N,N-dimethyl-1,3-thiazol-2-amine
N-ethyl-N-methyl-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridine-3-carboxamide
2-methoxy-1-[4-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]ethan-1-one
5-[1-(4-methylpyrimidine-5-carbonyl)pyrrolidin-2-yl]-N-(pyridin-2-yl)thiophene-2-carboxamide
2-[4-(5-chloropyridine-2-carbonyl)piperazin-1-yl]-1,3-benzothiazole
methyl 2-{[7-(pyridine-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}benzoate
1-(2-{[(4-ethylphenyl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2,4-dihydroxyphenyl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-4-(trifluoromethyl)benzamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-oxo-1,6-dihydropyridine-2-carboxamide
2-[(2-methoxypyrimidin-5-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-(2-hydroxyethyl)-8-(3-methoxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
cyclopentyl 4-{[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]amino}benzoate
4-benzyl-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
6-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-1-(propan-2-yl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
1-(4-{3-[({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(5S,9aS,9bS)-5-(3,7-dimethyl-1H-indol-2-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-[(2,3-difluorophenyl)methyl]-2-(ethanesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
4-(4-{1-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
4-methyl-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine
1-(4-fluorophenyl)-4-(furan-2-carbonyl)-1,4-diazepane
1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-(pyrrolidin-1-yl)piperidine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
methyl 1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
3-(3-chlorophenyl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1,2,4-oxadiazole
4-hydroxy-2-({methyl[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)quinoline-6-carboxamide
1-[2-(2H-1,3-benzodioxol-5-yl)phenyl]piperazine