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1-benzoyl-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]piperidin-4-amine
4-[(3-fluorophenyl)methyl]-1-[(2-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-[4-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
2-[4-(methylsulfanyl)phenyl]-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]acetamide
1-methyl-4-{[4-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}piperazine
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxamide
1-(2,6-diaminopyrimidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(4-ethylphenyl)ethyl]amine
2-ethyl-6-methyl-4-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
4-[(4-fluorophenyl)methyl]-1-(5-fluoropyrimidin-2-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-(carbamoylmethyl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]piperidine-3-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
1-methyl-N,N-bis(pyridin-3-ylmethyl)azepane-2-carboxamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]benzamide
(1S,6R)-9-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(2S)-2-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-phenylpropanamide
[(5-ethylpyridin-2-yl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
methyl (1R,3R,3aR,6aS)-5-methyl-4,6-dioxo-3-[(E)-2-phenylethenyl]-1-(propan-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-({5-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[(2-methylphenyl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
9-cyclopropanecarbonyl-2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecane
5-[(1R,4S)-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
1-cyclopentyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
5-ethyl-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
2-(4-fluorophenyl)-N-(2-{7-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-indole
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
N-cyclopentyl-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-methyl-1-benzofuran-7-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(2-methyl-1H-imidazol-1-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]propanamide
4-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1-ethyl-1,2-dihydropyridin-2-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-1,4-diazepan-5-one
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}-4-methylpiperazine
6-butyl-2-{4-[(4-fluoropiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
(4aR,6R,8aS)-2-[(3-fluorophenyl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-{3-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}acetamide
3-{1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]piperidin-4-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-({2-[cyclopentyl(methyl)amino]ethyl}(methyl)sulfamoyl)-N-ethyl-N-methylbenzamide
2-(5-ethyl-1-benzofuran-3-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-{[2-(4-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
methyl 2-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-3-hydroxypropanoate
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-N-(2-phenylethyl)piperidine-4-carboxamide
7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-6-(furan-2-yl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
3-chloro-N-cyclopentyl-4-{[1-(4,4,4-trifluorobutan-2-yl)piperidin-4-yl]oxy}benzamide
1-(2-propyl-1,3-thiazole-4-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-{2-benzyl-7-[4-hydroxy-4-(pyridin-2-yl)piperidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-5-yl}propanamide