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4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(2-phenylethyl)morpholine
4-(2,2-dimethylpropyl)-3-{2-[4-(3-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-(3-fluorophenyl)-6-[(1-methyl-1H-indol-3-yl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
(1R,2S)-N1-butyl-N2-[(5-chlorothiophen-2-yl)methyl]cyclohexane-1,2-dicarboxamide
4-[2-(1H-imidazol-1-yl)ethyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-(1,3-benzothiazol-2-yl)-4-(3-methoxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2R)-2-amino-3-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
N-[1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
({4-cyclopropyl-5-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-chloro-N-(2-methoxyethyl)-4-[(1-methylpiperidin-4-yl)oxy]benzamide
1'-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-chloro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
{1-[(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-cyclopropanecarbonyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
methyl 2-(7-chloro-3-{[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl}-2-oxo-1,2-dihydroquinolin-1-yl)acetate
ethyl 4-{1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(2H-indazol-2-yl)acetamide
1-cyclohexyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4-diazepane
8-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{4-[2-chloro-5-(trifluoromethoxy)phenyl]-1H-pyrrole-2-carbonyl}piperidine
1,1-dioxo-N-{2-[2-(pyridin-2-yl)ethoxy]phenyl}-1λ6-thiomorpholine-4-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-hydroxy-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
8-(3-methylpyrazin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[2-(2-methoxy-4-methylphenoxy)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
9-(cyclopropylmethyl)-4-[2-(1H-imidazol-1-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[3-(4-chloro-3-methylbenzoyl)-9-propyl-3,9-diazaspiro[5.5]undecan-1-yl]methanol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-ol
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
2-cyclopropyl-5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}pyrimidine
3-(4-fluorophenyl)-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1H-pyrazole-5-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1H-imidazol-2-ylmethyl)acetamide
2-amino-7-(3-methoxy-2-methylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[4-(hydroxymethyl)phenyl]-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-[bis(pyridin-3-ylmethyl)amino]-2-(5-fluoro-2-methoxyphenyl)acetic acid
(2S,4R)-N-ethyl-1-(2-hydroxybenzoyl)-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
4-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-(3-methoxypropyl)-5-{1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-benzoyl-1-[1-(4-fluorophenyl)pyrrolidin-3-yl]piperidine
2-({3-[(3,4-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1,3-thiazole
4-methoxy-N-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
ethyl 1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
2-acetyl-8-(5-acetylthiophene-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid