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(1s,4s)-4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]cyclohexan-1-ol
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methylpiperidine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
9-(5,6-dimethylpyridine-3-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-[(5-methylfuran-2-yl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
7-(5-chloropyridin-2-yl)-4-[2-(pyridin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(piperidin-1-yl)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
3-[5-(2,6-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]propane-1,2-diol
4-(1-benzyl-1H-imidazol-2-yl)-1-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidine
5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-(pyridin-2-yl)pyrimidine
N-[(4-chlorophenyl)methyl]-5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
benzyl({[3-(3-cyclohexylpyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl})methylamine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-ethyl-N-(oxan-4-ylmethyl)-2-(2-oxoazepan-1-yl)acetamide
N-(1-benzylpiperidin-4-yl)-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-[(2,3,6-trifluorophenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(piperidin-1-ylmethyl)benzamide
3,5-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,2-oxazole-4-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
2-[4-(3-benzoylpiperidin-1-yl)piperidine-1-carbonyl]pyrazine
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2,5-dimethyl-1,3-oxazole-4-carboxamide
5-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
2-(2-hydroxyethyl)-6-[4-(1H-pyrazol-3-yl)benzoyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-2-phenyl-1,3-oxazole
8-(5-methylpyridine-3-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-benzamido-5-{[(2-methylphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(4-fluorophenyl)-1,4-diazepane
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
ethyl 5-(2H-1,3-benzodioxole-5-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3S,5R,9R)-N-(2,4-dichlorophenyl)-5-hydroxy-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxamide
3-[3-chloro-4-(propan-2-yloxy)phenyl]-1-[(5-methylpyrazin-2-yl)methyl]urea
3-{2-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-1,3-oxazolidin-2-one
4-(dimethylamino)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)butanamide
methyl 2-({5-[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-2-yl]thiophen-2-yl}formamido)acetate
(4aS,7aR)-1-(2-hydroxyacetyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}-N-methyloxolan-3-amine
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-(4-{1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}thiophen-2-yl)ethan-1-one
2-(2-cyclopropylacetyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-(methylsulfanyl)propyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-cyclopropyl-N-[(2,3-difluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]morpholine-2-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,3-dimethylfuran-2-carboxamide
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
[(5-ethylfuran-2-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
7-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(methylsulfanyl)propan-1-one
4-ethyl-3-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(propan-2-yl)pyrimidine