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N-cyclopropyl-2-[4-({[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]carbamoyl}amino)phenyl]acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1S,9S)-11-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-({4-[5-(2-chlorophenyl)furan-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
1'-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-({2-[2-(2,5-dimethylphenyl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,4-triazole
3,7-dimethyl-11-[(2,4,6-trimethoxyphenyl)methyl]-3,7,11-triazaspiro[5.6]dodecane
4-[({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-2,6-dimethylphenyl acetate
3-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
3-(piperidin-3-yl)-N-[(4-sulfamoylphenyl)methyl]benzamide
2-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-2-azaspiro[4.5]decan-3-one
N-[4-(oxolan-2-yl)butyl]-2-[(prop-2-en-1-yl)amino]benzamide
(2S,4R)-N-methyl-4-[4-(4-methylbenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
(3R,9aR)-3-(hydroxymethyl)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-methyl-1-[2-(3-methyl-3-phenylpiperidin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1,2-oxazol-3-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4S)-4-(cycloheptylamino)-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(4-chloro-2-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}phenoxy)acetamide
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-[(4-methylphenyl)methyl]-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-amino-6-(2,5-dichlorophenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
N-(4-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)benzenesulfonamide
(2S,4R)-1-(2-methylpropyl)-N-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-(1-benzofuran-2-ylmethyl)morpholine-2-carboxylic acid
2-({7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)benzonitrile
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-{3-[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
2-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)-1H-1,3-benzodiazole
N-cyclopentyl-N-[2-(dimethylamino)ethyl]-3-(pyridin-4-yl)propanamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
N-(1-benzylpyrrolidin-3-yl)-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-(oxan-4-yl)piperidin-3-amine
N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylpropanamide
N-[3-(methylsulfanyl)propyl]-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
3-[(4aR,7aS)-4-[3-(ethylsulfanyl)propanoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-[2-(2-fluoro-5-methoxyphenyl)phenyl]ethan-1-amine
5-(2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-cyclopropyl-N-(5-methyl-2-pentanamidophenyl)-1H-pyrazole-4-carboxamide
4-{1-[1-(3-fluorobenzoyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
5-[(benzyloxy)methyl]-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazole
1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(2-methoxyphenyl)-3-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
6-(3-chloro-2-fluorobenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
1-(3,5-dimethylphenyl)-4-(1H-indole-6-carbonyl)piperazin-2-one
2-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole