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2-(cyclopropylmethyl)-N-(2,6-dimethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-(4-methanesulfonylbenzoyl)-3-(1H-pyrazol-5-yl)piperidine
(1R,2S)-N-methyl-2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclohexane-1-carboxamide
N-cyclooctyl-5-(2-ethylpiperidine-1-carbonyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-(2-methoxyethyl)-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
3-(3-methoxyphenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
5-chloro-2-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-amino-6-tert-butyl-4-(dimethyl-1,2-oxazol-4-yl)pyridine-3-carbonitrile
3-oxo-N-[1-(pyrazin-2-yl)piperidin-3-yl]-3,4-dihydroquinoxaline-2-carboxamide
3-{2-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
4-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridine
3-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)pyridine
2-[4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
[(4-{2-[4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N,N-dimethylpyridin-2-amine
N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl][(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-(morpholin-4-yl)-2-(4-{[(quinolin-8-yl)amino]methyl}phenoxy)ethan-1-one
3-{[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}propane-1,2-diol
5-(4-acetylphenoxymethyl)-N-cyclohexyl-1,2-oxazole-3-carboxamide
2-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
4-(3-methyl-1-benzothiophene-2-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-(4-chlorophenyl)-4-[5-(piperidine-1-carbonyl)pyridin-2-yl]morpholine
(3S,5R,9R)-5-hydroxy-11-(naphthalene-1-carbonyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-(cyclohexylmethyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-6-oxopiperidine-3-carboxamide
N-[4-(8-hydroxyquinolin-2-yl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]propanamide
(3aS,6aS)-N,N-dimethyl-5-(5-phenoxyfuran-2-carbonyl)-octahydropyrrolo[3,4-b]pyrrole-1-carboxamide
1-benzyl-3-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]urea
(3S,4S)-1-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
[(3S,5R)-5-[(dimethylamino)methyl]-1-[3-(3-fluorophenyl)benzoyl]piperidin-3-yl]methanol
4-(2-fluorophenyl)-6-methylpyrimidin-2-amine
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-methylpyrazine-2-carboxamide
2-{8-[3-(furan-2-yl)benzoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
(4aS,8aR)-1-(4-hydroxybutyl)-6-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
1-[(1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
4-[(3R,5R)-5-[4-(5-methylpyrimidin-4-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
2,6-difluoro-4-methoxy-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-N-phenylpyrimidin-2-amine
4-[(4-methyl-5-{1-[3-(pyridin-3-yl)propyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-3-(pyridin-4-yl)propanamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-3-hydroxypiperidin-2-one
1-(oxolane-3-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
1-(2-chlorophenyl)-3-{1-[1-(thiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-methyl-8-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one