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3-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
N-{1-[1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
methyl 8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2-methoxyethyl)-N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-(1,3-dihydroxypropan-2-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(1H-indol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
2-(2,3-dihydro-1H-inden-1-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-6-carboxamide
methyl (2S,4S)-4-[(dimethylsulfamoyl)amino]-1-methylpyrrolidine-2-carboxylate
(2R,6R)-4-(dimethyl-1,3-thiazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
[1-(3-chloro-1H-indole-2-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
2-methyl-6-(piperidin-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidin-4-amine
N-[2-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)ethyl]pyridine-3-carboxamide
(2S,4S)-4-{4-[4-(2,5-dihydro-1H-pyrrol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
1-{2-[4-(3-phenylpropanoyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-methoxy-2-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenol
(1R,2R)-2-[ethyl({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)amino]cyclohexan-1-ol
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(dimethyl-1,3-thiazol-5-yl)-N-methylacetamide
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(2-methyl-1-benzofuran-5-yl)urea
N-{2-[2-(4-chlorophenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}morpholine-4-carboxamide
1-[4-({[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)thiophen-2-yl]ethan-1-one
N-[1-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-4-oxo-4-phenylbutanamide
{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})amine
1-{4-[(4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazin-1-yl}ethan-1-one
N-(naphthalen-2-yl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
2-amino-4-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}quinazoline-6-carboxylic acid
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
6-[(diethylamino)methyl]-N-[3-(1,3-oxazol-5-yl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[2-(butan-2-yloxy)phenyl]-3-[(6-hydroxypyrimidin-4-yl)methyl]urea
4-benzyl-3-ethyl-1-[(4-hydroxy-3-methylphenyl)methyl]-1,4-diazepan-5-one
N-butyl-N-cyclopentyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
1-[2-(4,4-difluoropiperidin-1-yl)-2-oxoethyl]-3-methyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-tert-butyl-3-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
1-(pyrazin-2-yl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
6-[2-(tert-butylsulfamoyl)phenyl]pyridine-2-carboxamide
8-(3-hydroxypropanoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
3-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-5-(propan-2-yl)-1,2-oxazole
7,7-dimethyl-2-(3-phenylpropyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]propanamide
5-(3,4-dimethoxyphenyl)-3-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
2-[2-({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[(2-methoxyphenyl)methyl]-1-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-3-yl]-3-methanesulfonylpropanamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-benzyl-N,N-dimethyl-5-{[2-methyl-2-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide