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[2-(azepan-1-yl)ethyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-methyl-2-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinazoline-4-carboxamide
(3S,4S)-4-(pyridin-2-yl)-1-[2-(2,2,6,6-tetramethylpiperidin-4-yl)acetyl]pyrrolidine-3-carboxylic acid
(3S,9R)-11-(naphthalene-1-carbonyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
3-[3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)phenyl]-N-methylpropanamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
methyl (2S,4S)-1-methyl-4-[4-(1H-pyrazol-1-yl)benzenesulfonamido]pyrrolidine-2-carboxylate
N-[(2,3-dimethoxyphenyl)methyl]-1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-amine
1-(6-methoxy-4-methylquinazolin-2-yl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]pyrrolidine-2-carboxamide
N-benzyl-3-[(cyclopentylamino)methyl]-N-methylpyridin-2-amine
N-methyl-5-(1-{2-[(prop-2-en-1-yl)amino]benzoyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N,N-dimethyl-7-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
5-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-4-propylpyrimidine
4-(carbamoylmethoxy)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
2-{2-[3-(3-methoxypropyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
5-methyl-1-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
3-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
3-phenyl-1-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]piperidine
5-(2-methylfuran-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3R,4R)-4-amino-1-[3-(3-methoxyphenyl)benzoyl]piperidin-3-ol
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
2,5-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)propanamide
8-(2-aminoacetyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cycloheptanecarbonyl-4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine
8-[2-(azepan-1-yl)acetyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-phenylpropyl)-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,4-diazepane
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
7-fluoro-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methylquinoline-4-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
4-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
1-phenoxy-2-{4-[(2,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-6-(methoxymethyl)pyrimidin-4-amine
1-methyl-8-({4-[methyl(phenyl)amino]phenyl}methyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-dihydrophthalazin-1-one
3-(1,2-oxazinan-2-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
4-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)morpholine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-hydroxyethan-1-one
N-cyclopentyl-3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]benzene-1-sulfonamide
2-ethyl-4-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1,3-thiazole-5-carboxamide
1-(4-ethylpiperazin-1-yl)-3-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-ethylpiperidin-3-ol
5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(4aS,8aS)-2-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-7-propyl-decahydro-2,7-naphthyridin-4a-ol
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
1-[(2,6-difluorophenyl)methyl]-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 5-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2,4-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid