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6-methyl-2-[1-(4-methylpiperazine-1-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(1S,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N,4-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}pyrimidin-2-amine
1-(2-methoxyphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(pyridin-4-ylsulfanyl)acetamide
N-(1-hydroxy-2-methylpropan-2-yl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(3-methylpyridin-2-yl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazine
(4aS,7aR)-1-(oxane-4-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
5-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
4-{[1-(cyclohexylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}-3,3-dimethylpiperazin-2-one
4-ethyl-3-{1-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,4S)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-benzyl-3-ethyl-1-(4-hydroxy-3-methylbenzoyl)-1,4-diazepan-5-one
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
2-(4-ethylpiperazin-1-yl)-N-[2-(2-fluorophenyl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-tert-butyl-4-({[4-(dimethylamino)-5-methylpyrimidin-2-yl](methyl)amino}methyl)pyrrolidin-2-one
1-tert-butyl-N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide
3-(2,4-dimethoxyphenyl)-5-[1-(1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazole
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-{4-[(2-methylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
(3R,4S)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
(1S,4S)-2-(3-chlorophenyl)-5-(quinolin-6-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(4-methylphenoxy)ethan-1-one
[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
3-(1H-1,3-benzodiazol-2-yl)-N-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]azetidine-1-carboxamide
N-ethyl-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
5-acetyl-N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2,7,8-trimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
2-{9-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(3R,4R)-3-hydroxy-N-(2-methylphenyl)-4-{[(3-methylpyridin-2-yl)methyl]amino}pyrrolidine-1-carboxamide
3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
1-[(2,3-difluorophenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
3-(2-amino-1,3-thiazol-4-yl)-1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]propan-1-one
2-(dimethyl-1,3-thiazol-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
1-(3-cyclopropylpropanoyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
4-ethyl-3-(2-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)piperazin-2-one
2-chloro-N-{[1-(4-ethylbenzenesulfonyl)piperidin-3-yl]methyl}benzamide
N-ethyl-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-(pyridin-4-ylmethyl)acetamide
7-(5-methylthiophen-2-yl)-4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-(quinolin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1R,5R)-6-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-{[(1H-indol-4-ylmethyl)(methyl)amino]methyl}-1-methylpyrrolidin-2-one
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(cyclopropylmethyl)acetamide