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N-({1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}methyl)furan-2-carboxamide
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-2-{3-methyl-2-oxo-2H,3H-imidazo[1,2-a]pyridin-3-yl}acetamide
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-ethoxyphenyl)piperazine
1-(cyclohex-3-en-1-ylmethyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
6-(3-hydroxypiperidin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
(2S,4S)-1-{[4-(methylsulfanyl)phenyl]methyl}-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
1-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
4-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-5-benzyl-2-methylpyrimidine
3-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]benzoic acid
3-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-(pyrimidin-4-ylmethyl)benzamide
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
methyl 4-{5-chloro-2-[(2-cyclopropylacetamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-imidazol-2-yl]-5-ethylpyridine
1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-methoxy-N-[3-methyl-1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)butyl]acetamide
N,N-diethyl-1-(1-propylpiperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
8-cyclobutanecarbonyl-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(4aS,8aS)-2-{[2-methyl-5-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
2-(2-hydroxyethyl)-9-[6-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(2S)-2-amino-4-(methylsulfanyl)-N-[3-(2-phenylacetamido)phenyl]butanamide
5-benzyl-3-(pyridin-3-ylmethyl)-5-[1-(thiolan-3-yl)piperidin-4-yl]imidazolidine-2,4-dione
N-(2,3-dihydro-1H-inden-4-yl)-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
2-(2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
5-(2,6-difluoro-3-methylphenoxymethyl)-3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazole
9-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(8-methoxy-2H-chromen-3-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
methyl 6-[(2,4-dimethylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-phenyl-N-(1H-1,2,4-triazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-5-propyl-1,2-oxazole-3-carboxamide
3-(propan-2-yl)-5-(1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}pyrrolidin-2-yl)-1,2,4-oxadiazole
(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethyl-N-[4-(trifluoromethyl)phenyl]piperidine-1-carboxamide
3-methyl-6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyridazine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}quinoline-3-carboxamide
N-[(2S)-1-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](2-methylpropyl)amine
N-(3-fluorophenyl)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperidin-3-amine
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
1-[3-(2-methoxyphenyl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
6-methoxy-3-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-benzofuran-2-carboxamide
2-amino-6-cyclopropanecarbonyl-4-(3-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-[3-(hydroxymethyl)phenyl]acetic acid
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(4-fluorophenoxy)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(piperidin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
7-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide