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2-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}quinoline
2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(3-cyano-4-methylphenyl)-3-(3-ethylphenoxy)azetidine-1-carboxamide
5-(methoxymethyl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}furan-2-carboxamide
1-cycloheptyl-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
methyl 4-{[(2S,4R)-2-[(2-methyl-1,3-benzothiazol-5-yl)carbamoyl]-4-(pyridin-2-ylsulfanyl)pyrrolidin-1-yl]methyl}benzoate
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-6-methoxypyrimidin-4-amine
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2-methoxyethyl)-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
2-({2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1-(4-methoxy-3,5-dimethylphenyl)urea
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-(2-fluorophenyl)benzoyl]pyrrolidin-3-yl]methanol
1-{2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
N-{3-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
1-methanesulfonyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidin-4-amine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-{1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
2-[(3,4-dimethylphenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(cyclohex-3-en-1-ylmethyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,1-dimethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-fluoro-3-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,4-dihydroquinolin-4-one
1-(pyridin-2-ylmethyl)-4-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-diazepane
3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
N-cyclopropyl-3-{[(4-ethyl-1,3-thiazol-2-yl)methyl]sulfamoyl}benzamide
4-chloro-3-({[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-(1H-pyrazol-5-yl)piperidine
3-({1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
N-[2-fluoro-3-(trifluoromethyl)phenyl]-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
1-[2-({thieno[2,3-d]pyrimidin-4-yl}amino)ethyl]piperidine-3-carboxamide
3-({4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-5-methoxy-1H-indazole
2-{3-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]piperidin-1-yl}acetamide
{3-[(3-methoxyphenyl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}methanol
4-(5-methylpyridin-2-yl)-1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-4-ol
(4aS,8aR)-6-(3,6-dimethylpyrazin-2-yl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-methyl-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
N-[(3R,4S)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
(4aS,7aR)-1-[(4-ethoxyphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-butyl-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(2-fluoroethyl)-2-{4-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]morpholin-3-yl}acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
1-[1-(6-{[2-(1H-imidazol-2-yl)ethyl]amino}pyridine-3-carbonyl)piperidin-3-yl]-3-methylbutan-1-one
(1R,2S,6R,7S)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-azatricyclo[5.2.2.02,6]undecane
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(2-methoxyethyl)pyridin-2-amine
4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
(2S)-2-amino-3-hydroxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea