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2-ethyl-5-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrimidine
7-chloro-3,5-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
3-(3-chlorobenzoyl)-1-(2,3-dihydro-1H-inden-2-yl)piperidine
[3-(3-methoxypropyl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-3-yl]methanol
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxylic acid
[2-(diethylamino)ethyl]({[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
1-(pent-2-yn-1-yl)-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-hydroxy-2-methylpropan-2-yl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]imidazolidin-2-one
methyl 6-(4-methylpentanoyl)-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
9-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 5-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-5-oxopentanoate
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-2-yl]propan-1-ol
2-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1-benzofuran-5-carboxamide
(3R,4S)-4-{4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
3-(1,2-oxazinan-2-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanamide
(2S,4R)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
3-[5-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]benzoic acid
(benzylsulfamoyl)({2-[(dimethylamino)methyl]phenyl}methyl)methylamine
(3aS,6aS)-2-cyclobutanecarbonyl-5-(1,3-thiazol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-phenylpropan-1-one
5-{1H-pyrazolo[3,4-b]pyridin-1-yl}pyridin-2-amine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
3-({2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-2-(thiophen-3-ylmethyl)propan-1-ol
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
2-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
2-amino-5-ethyl-4-(4-methanesulfonylphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
(1S,5R)-3-(1-ethyl-1H-indole-5-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4-chloro-2-methylphenyl)-3-cyclopropyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,3R,6R)-5-{imidazo[1,2-a]pyridine-2-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-methylphenyl)-3-{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
1-(cyclohexylmethyl)-N-methyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
7-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-benzyl-8-(3-ethyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecane
N4-cyclobutyl-N2-cyclopropyl-7-(1H-imidazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-4-carboxamide
2-(3-fluorophenyl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-5-carboxamide
1-{4-methyl-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-5-yl}ethan-1-one
3-[2-(2-methyl-5-oxo-4-phenylpiperazin-1-yl)-2-oxoethyl]-2,3-dihydro-1,3-benzoxazol-2-one
2-[4-(3-phenoxypropyl)piperazin-1-yl]ethan-1-ol
N-[(3R,4S)-4-propyl-1-(pyrimidin-2-yl)pyrrolidin-3-yl]morpholine-4-sulfonamide
4-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
(2E)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-3-phenylprop-2-enamide
2-(3,4-dimethoxyphenyl)-5-fluoro-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole