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3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]urea
(2R,3S,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(4,4,4-trifluorobutanoyl)-1,4-diazepan-2-one
4-chloro-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1-methyl-1H-indazole
6-(1-{2-amino-6-[(4-methylphenyl)sulfanyl]pyrimidin-4-yl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
8-(1-benzofuran-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[(E)-2-phenylethenyl]-1,3-benzoxazole
5-[3-(benzyloxy)piperidine-1-carbonyl]-4-phenylpyrimidin-2-amine
9-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
6-(1H-indol-5-yl)-N,N-dimethylpyridazin-3-amine
3-[2-(2,2-dimethylpiperazin-1-yl)-2-oxoethyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
5-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2-propylpyrimidine
3-(dimethyl-1,2-oxazol-4-yl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
2,4-dichloro-3-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenol
1-[(2,6-difluorophenyl)methyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
3-methoxy-N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2H-1,3-benzodioxole-5-carboxamide
4-{[1-(2-hydroxybenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-ethyl-4-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)pyrrolidin-2-one
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(4-hydroxyphenyl)ethan-1-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4,6-dimethoxypyrimidine
(1S,5R)-6-(1-methyl-1H-pyrazole-4-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S)-4-methyl-1-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-2-phenylpiperazine
4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
N-[2-(3-methoxy-4-propoxyphenyl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
6-ethoxy-3-[(4-hydroxypiperidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
3-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
2-({4-[3-(3,4-dimethoxyphenyl)propanoyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
2-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)pyridine
9-[2-(2-ethylphenoxy)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
2-(2-methoxyphenyl)-5-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}pyrimidine
4-fluoro-N-[3-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]benzene-1-sulfonamide
3-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methoxy)phenol
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-pyrazole-4-carboxamide
4-ethyl-3-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4-acetyl-4-phenylpiperidin-1-yl)-2-oxoethyl]benzamide
2-{5-[1-(2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
7-methoxy-3-[4-(4-methylpiperazin-1-yl)benzoyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
4-methyl-2-(propan-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,3-thiazole-5-carboxamide
1-cyclopentyl-4-[({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
1-{4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
3-{1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-N-(propan-2-yl)-2-(thiophen-2-yl)acetamide
1-{4-[(3-methoxy-2,2-dimethylpropyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one